Ahụ ike, Preparations
"Disulfiram": reviews. "Disulfiram": nkọwa, price
N'isiokwu a, anyị kpebiri na-agwa gị na nke a bụ ọgwụ dị ka "Disulfiram". Ntuziaka maka ojiji, nzaghachi na-egosi nke ego a ga-kọwara n'okpuru ebe a. Ke adianade do, ị ga-amụta na ihe ndị na-eri si ọgwụ, ọ na-emepụta na ihe ọ bụla n'ụdị na a gụnyere na ya mejupụtara, na na. D.
The ụdị na mejupụtara nke nkwakọ
The agwọ ọrịa "Disulfiram", ntuziaka maka ojiji nke a na-nchọ na a igbe mere nke katọn, ahịa na ụdị mmanu mmanu ngwọta na mbadamba maka onu nlekọta na nkunye.
The mbụ n'ụdị na-emepụta na vials nke 20 ml, na abụọ na nke atọ - na iko ite na 10 na 20 nkeji karị.
The n'ọrụ mgwa nke agwọ ọrịa bụ disulfiram. E wezụga ya, ọgwụ nwere nwekwara mmiri (dabere na ntọhapụ forms): sodium chloride, mannitol, starch, sodium stearate, mkpọ-6000, MCC, calcium diphosphate, hydroxypropyl cellulose, stearic acid na polyoxyl 40.
pharmacological Njirimara
Gịnị bụ tupu anyị na nkà mmụta ọgwụ? Ihe ha na-ekwu banyere ya ọgwụ reviews? "Disulfiram" nwere a akpọ mgbochi mmanya mmetụta.
Mgbe ị na-enweta ngwá ọrụ a na-ama maka ya ịrịba mmetụta na mmanya metabolism. N'ihi ya, mma metabolites na-guzobere, nke dịkwuo ịta nke nsi dị ka acetaldehyde. Ọ bụ ya na-ekpebi ịdị irè nke ọgwụ.
Na igba ogwu n'akwara ochichi nke a agwọ ọrịa, nakwa dị ka ya onu ọrịa fọrọ nke nta ozugbo amalite na-eche na-ekpo ọkụ flushes, nnukwu dyspepsia, tachycardia, asthenia ike na ọbụna na-eyi egwu hypotension. Ke adianade do, ọdịdị nke igbu egbu site acetaldehyde eme mkporomaasi ka mmanya na mkpochapu ndidi nzube mmanya.
pharmacokinetic parameters
Gịnị echiche nwere ọgwụ kinetic kwa? Gịnị banyere ya absorption akụkọ reviews? "Disulfiram" nnọọ ngwa ngwa na fọrọ nke nta kpamkpam etinye obi gị dum na gootu.
Mgbe na-eji ya, e nwere a elu metabolism nke nọ n'ọrụ akụrụngwa, n'oge nke ọtụtụ metabolites kpụrụ. Nweta nke ngwaahịa a rụrụ site na akpa ume na-na akụrụ.
egosi
Drug "Disulfiram", ego nke nke na-egosi n'okpuru, gosiri maka:
- ọgwụgwọ nke ala ala aṅụrụma;
- mgbochi nke nlọghachi azụ na ọgwụgwọ nke ala ala aṅụrụma.
Were a ọgwụ na ya ezi uche ekwesighi. Ọ ga-ahọpụta a dọkịta.
contraindications
Drug "Disulfiram" intravenously na ọnụ na-adịghị akwadoro maka ndị na-esonụ ọrịa:
- neuropsychiatric ọrịa;
- akwụkwụ na-adọ;
- arịa ọrịa shuga.
Ọzọkwa, a ọgwụ na-adịghị gosiri n'oge ime, na uche na-arụsi ọrụ ike akụrụngwa na onye ọzọ na akụrụngwa, ara.
Anyị ga na-ekwukwa na ihe ókè ịkpachara anya a ọgwụ na-atụ aro iji na-ọrịa na mkpọchị imeju ọrụ, akụkụ okuku ume na usoro na akụrụ.
Drug "Disulfiram": ntuziaka maka ojiji
The ojiji nke ọ bụla n'ụdị nke ego bụ ime na na dọkịta iwu. The dọkịta na iwu ji na-akpa àgwà a full ule onye ọrịa, na mgbe ahụ họrọ otu onye ọgwụgwọ Usoro na dose maka ya.
Dị ka ntụziaka, nkezi kwa ụbọchị dose nke ọgwụ maka onu ochichi bụ banyere 125-500 mg.
Ma ihe ndị ọgwụ na nkunye nke ọgwụ, mgbe ahụ, a na usoro ga-rụrụ site ahụmahụ ẹkesikpede. Na nke a na-atụ aro usoro onunu ogwu nke ọgwụ na-adabere na àgwà nke ndidi na ogo nke ẹdude ọrịa.
mmetụta
mmetụta nke ọgwụ ahụ na ajụjụ nwere ike m na-akpọ? Gịnị banyere nke a na-ekwu na reviews? "Disulfiram" adịkarịghị ibu akpata ize ndụ n'akụkụ Jeremaya mere. Mgbe ingested o nwere ike ịbụ na ụfọdụ ndiiche na digestive tract na ọnụnọ nke dara uto na mmepe nke ịba ọcha n'anya.
Ke adianade do, imebi nwere ike ime na ụjọ usoro ọrụ. Ndị dị otú ahụ adịghị mma na ọnọdụ na-agụnye polyneuritis nke ala ụkwụ, ọrịa uche, ebe nchekwa ọnwụ, mgbagwoju anya na isi ọwụwa.
Ọzọkwa, adịghị ewepu na mmepe nke dị iche iche nfụkasị Jeremaya mere, nke na-triggered site na mmanya na-egbu (e.g., ida, ọrịa strok, gbasara obi arrhythmias, ọrịa ụbụrụ edema na myocardial infarction).
Mgbaàmà nke ovadozu
Nkwadebe "Disulfiram" na elu doses nwere ike ime ka mmetụta dị otú ahụ dị ka ida, amaghị onwe na ize ndụ akwara ozi Jeremaya mere.
Iji kpochapụ ndị a mgbaàmà kwesịrị iwepụta symptomatic ọgwụ n'ụlọ ọgwụ, nke ga-abụrụ na-agụnye detoxification eme.
mgbochi agwọ ọrịa
Ọkachamara gaara egosi na zuru ezu neutralization nke ọgwụ ike-atụle.
Ọ bụrụ na ọ dị mkpa, na mmepụta "Disulfiram" si ahụ mmadụ (e.g., na oké Jeremaya mere ka ọhụrụ nakweere dose mmanya) a rụrụ ụfọdụ usoro.
Dị ka ihe ngwọta nke a iji ọgwụ ọjọọ eme ascorbic acid. Ọ na-ndinọ intravenously. Nke a mmewere adịghị ekwe ka mmanya ghọọ acetaldehyde, nke na, n'eziokwu, na-akpata ahụ erughị ala.
Ha pụkwara eji ephedrine na H1-blockers.
ọgwụ interactions
Ọ dị mma iji ọgwụ ọjọọ ndị ọzọ tupu anyị na nkà mmụta ọgwụ? Gịnị banyere ndị ọgwụ ọjọọ interactions reviews na-ekwu? "Disulfiram" na Nchikota na anticoagulants enwekwu ha ihe, ma na-enwekwu ihe ize ndụ nke ọbara ọgbụgba.
Imekotaotuugbo ọgwụgwọ na ọgwụ ọgwụ nke na-metabolized na imeju, nwere ike budata ịkparị n'oge usoro.
Na ijikọta Mao inhibitors, tricyclic antidepressants na phenothiazine nkwekọrịta na "Disulfiram" nwere ike na-eme ka ntoputa nke mgbagwoju n'akụkụ Jeremaya mere.
The Nchikota nke a pụtara na "buspirone" na-akpata mmepe nke nkwenkwe ụgha. Ndị dị otú ahụ na nkà mmụta ọgwụ dị ka "Amitriptyline", mgbe mgbe, enhances mmetụta nke "Disulfiram" na-akpọlite ya na-egbu egbu mmetụta na ụjọ usoro.
E lee ya anya agwọ ọrịa ike nke na-amụba ịta nke chlordiazepoxide na diazepam n'ime ọbara, na-ebelata ike nke na-egbu egbu Jeremaya mere na-eme ka dizziness.
Na Nchikota "Disulfiram" na "isoniazid" nwere ike ịzụlite ịda mbà n'obi na dizziness, "metronidazole" - mgbagwoju anya na nnukwu psychosis, a "Omeprazole" - isi nsụhọ, na caffeine - belata ya excretion si ahụ.
"Chlorzoxazone" enwekwu ịta nke mgbochi mmanya ọgwụ na ọbara, na "Chlorpromazine" amplifies hypotension.
Drug "Disulfiram": reviews, price na analogues
Yiri mmetụta nwere ọgwụ ọjọọ ndị dị ka "Ekzorran", "Radotera", "Aspen", "Krotenal", "Tetlong", "Refuzal", "Stoptil", "Antietil", "Kontrapot", "Tetradin", "Antietan" "Dizetil", "Alkofobin", "Aversan", "Anticoli", "Antabuse", "Esperal", "Lidevin", "Abstinil".
Ego ole ka a ọgwụ ọjọọ, "Disulfiram"? The price nke a ọgwụ na mbadamba àmà 200-1000 rubles (dabere na emeputa). Banyere ịkụbanye udi, nakwa dị ka mmanu mmanu solution, ha nwere ike zụrụ maka 600-2400 rubles.
Kasị reviews nke ugbu Nwa na-nti. Ọ bụ ihe kwesịrị ịrịba ama na a ọgwụ a na-eji maka na nzuzo ọgwụgwọ nke ndị mmadụ na aṅụrụma. Ndị ọkachamara na-adịghị ike ikwu na-enye nke a owuwu enweghị onye ọrịa ahụ ihe ọmụma.
Dị ka nzaghachi nke ndị na-eji ọgwụ ọjọọ na-ewere ya nnọọ irè ọgụ agụụ na-a ọhụrụ dose mmanya. A, mgbe na-anata ọgwụ na onye ọrịa na-ebilite mkporomaasi ka mmanya. Ọ bụrụ na onye aṅụrụma onunu e gafere mgbe iji ọgwụ, ọ na-akpata nnukwu dyspepsia, flushing, oké asthenia, tachycardia, na ọbụna na-eyi egwu hypotension.
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