Ahụ ike, Preparations
Drug "varenicline". ntụziaka
Drug "varenicline" na-akpan iji German na-emepụta ọgwụ na ụlọ ọrụ Pfizer ọgwụ na e mere na-enyere na-ese siga na-alụso nicotine riri ahụ. Na pharmacies, ọgwụ nwere ike zụrụ n'ụdị film-ntekwasa mbadamba.
Drug "varenicline" ntụziaka nke na-atụ aro na ọ dị ka a na ụgbọala e mere n'ihi na ise siga cessation okenye, na-emi esịnede nke ugbu a mmewere nke varenicline. Inyeaka mmiri na isi mbadamba bụ: microcrystalline cellulose, anhydrous calcium hydrogen phosphate, croscarmellose sodium, colloidal sịlịkọn dioxide na magnesium stearate. Na shei nke usoro onunu ogwu ụdị mejupụtara titanium dioxide, polyethylene dị iche iche e ji esiji ákwà.
Drug "varenicline" ntụziaka nke na-akọwa n'ụzọ zuru ezu na ya pharmacological Njirimara, na-akpa ya mgbochi-ise siga edinam site Isi nọ n'ọrụ mgwa. Ọtụtụ ndị ọkà mmụta sayensị ọmụmụ gosiri na ntọhapụ nke dopamine na ahu na mmetụta nke obi ụtọ site a sịga na-esi mmetụta nke nicotine na nicotine anabata emi odude ke Central ụjọ usoro.
Vareniks-arụpụta ihe mmetụta nke bụ zuru ezu iji belata mgbaàmà nke ịkwụsị ịṅụ sịga na mbenata agụụ a sịga. Nke a na umi nwere emegide ọrụ, adịghị ekwe ka nicotine kpọtụụrụ na CNS anabata. N'ihi ya, onye ọrịa nwere dịghị riri obi ụtọ nke na-aṅụ sịga, na-ebelata ihe mgbaàmà nke agụụ maka ise siga. Vareniks, abanye na-ese siga, na-emeghachi omume na otu ụbụrụ anabata dị ka nicotine. Na nke a, ntọhapụ nke dopamine na-emepụta na nta quantities. N'ihi ya, mgbe eji ọgwụ na-anapụta a mmetụta nke obi ụtọ, yiri mmetụta nke nicotine na ahu na onye na-adịghị ike ahụ erughị ala mgbe enye elu sịga. Ọzọkwa, ọgwụ nkanka na nicotinic anabata maka ụtaba. Nke a usoro blunts obi ụtọ nke na-ese sịga.
Nkwadebe "varenicline" ntụziaka nke na-enye nkọwa nke usoro nke ya ochichi, pụtara maka anụ ụlọ iji. Na-atụ aro dose akụrụngwa nke otu milligram nke varenicline ugboro abụọ kwa ụbọchị ruo ụbọchị asaa mgbe titration.
Abụkarị ọgwụ "varenicline" ọgwụgwọ nke a na-kenyere a ọkachamara, na-a oge nke iri na abụọ izu. Tupu ịmalite iji ọgwụ na-kenyere a kpọmkwem ụbọchị mgbe ọ bụ zuru ojuju nke nicotine. Ọ bụ na-emekarị na nso nke asatọ iri na anọ na ụbọchị site ná mmalite nke ọgwụgwọ. Iji nweta ihe ịga nke ọma n'ihi ọrịa ga-kwadebere na uche. O kwesịrị agbamume na mkpali. Mgbe ọma ịlụ Bibie nicotine riri ọkachamara nwere ike ikwu na a yiri N'ezie nke na-ewere ndị ọzọ ọgwụ.
Drug "varenicline" (ntuziaka adọ aka ná ntị nke mmetụta na-ekwe omume n'oge ọgwụgwọ) nwere ike ime ka na-akwụsị akwụsị isi ọwụwa na ọgbụgbọ ma ọ bụ vomiting. Ọzọkwa yiri ka na-ehi ụra ọrịa na ehighị ụra nke ọma. Ọrịa ndị na-sonso anabata ndị erughị ala nke na-adịghị mma mmetụta nwere ike na-a nta dose nke ọgwụ. Ọ nwere ọgwụ ọjọọ, "varenicline" contraindications. Ọ na-adịghị ndinọ ka ọrịa iri na asatọ afọ, ime, lactating inyom, nakwa dị ka ụba uche na varenicline ma ọ bụ ihe ọ bụla nke excipients.
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