Ahụ ike, Preparations
"Izoket" Ịgba: ntụziaka ntuziaka, reviews, nkọwa, analogues, price
Taa, ọtụtụ ndị ọkachamara na nye iwu ka ọrịa vasodilator ịgba "Izoket" prophylactically ma ọ bụ, ma ọ bụrụ na ọ dị mkpa, cupping apịpịa.
pharmacology
Active gị n'ụlọnga nke ọgwụ rịaworo pectoris ji akpọ vasodilating na vasodilator Njirimara. Isosorbide dinitrate akpali guzobere nitrogen oxide na organism ma na-ebelata ihe ndị a chọrọ nke obi muscle nke oxygen na ume, si otú mbenata ibu na myocardium. Ọ n'ụzọ dị irè na-ebelata nsogbu na akpa ume mgbasa, mbelata ọbara-nri atrium, ebelata gbasara obi ventricular mgbidi erughị ala na decreasing diastolic nsogbu na systolic ọrụ rụọ ha. The ọgwụ nwere dịghị mmetụta ugboro nke contractions obi na gbatịrị ọma ụbụrụ arịa. Ọ nwekwara ike dịkwuo ọbara arịa nke Dura mater nke ụbụrụ na otú mwute na isi.
Ịgba "Izoket" ngwa ngwa etinye obi gị dum gafee mucosa nke ebe ọnụ, ya mere, mmetụta nke ya ngwa-amalite mgbe 30 sekọnd na dịruru ruo 120 nkeji. N'ihi ọsọ ọ na-emekarị kenyere ọrịa ozugbo enyemaka nke nnukwu ọnọdụ.
ntọhapụ Ụdị
The ọgwụ bụ ihe doro anya ihe ngwọta, nke bụ colorless na nwere onye aṅụrụma ísì ụtọ. Ọ na-abịa na abụọ iche:
- Ịgba "Izoket" na sublingual onunu ogwu. Na otu click na dispenser tọhapụrụ n'ụdị obere tụlee nke onye nke ya dose nke na-emi esịnede 1.25 mg nke nọ n'ọrụ mgwa - isosorbide dinitrate na inyeaka ọcha: ethanol na Macrogol 400. The aerosol mejupụtara ka a freon, Otú ọ dị ya na-akọ ọgwụ ọjọọ na-adịghị emerụ maka gburugburu ebe obibi. Emepụta uzo karama nke 15 ml, juru n'ọnụ na a igbe na a dispenser na ntụziaka. Glass karama maka 300 clicks (doses), na-enye ohere ka i nyochaa ego nke ọgwụ ọjọọ na-enweta a nnọchi na a-adọ ha n'ụzọ.
- The ngwọta na uche n'ụdị zubere maka infusions. 1 ml nke a nkwadebe ẹdude 1 mg nke nọ n'ọrụ mmewere nke isosorbide dinitrate na inyeaka bekee: sodium chloride, sodium hydroxide, mmiri. Otu mkpọ - 10 ml nke ngwọta maka infusion. Dị na katọn Ukwu nke 10 mbak ọ bụla.
egosi
Ịgba "Izoket" họpụtara ndị ọkachamara na stenokardicheskie ọgụ ụdị nile na dị ka a mgbochi ụfọdụ izere ha. Ọ na-atụ aro maka post-infarction states, myocardial infarction na nnukwu ogbo, na-amụba ndidi na IMS na ọgwụ nke akwara akwara spasm. Aerosol "Izoket" ọma ji dị ka a ọgwụ n'ihi na obi ọdịda ekpe ventricle.
- ejighị n'aka rịaworo aa na preinfarction ọnọdụ ma ọ bụ gara aga myocardial infarction;
- vasospastic rịaworo;
- myocardial infarction na nnukwu ụdị, mere site na odida nke ekpe ventricle nke obi;
- akwara vasospasm n'oge awa ahụ adọ;
- obi odida nke nile di iche iche;
- nnukwu ekpe ventricular obi odida;
- akpa ume edema.
Ụzọ nke ojiji nke aerosol
A nkwadebe n'ụdị a ịgba sprayed n'ime onu oghere onye ọrịa, n'ihi na nke a na ọ ngwa ngwa abatakwa ọbara iyi. Onye ọ bụla ọgwụ na-enye otu ingestion dose. Ntuziaka maka ojiji na-ezo aka n'ụzọ dị iche iche nke na-eji ọgwụ ọjọọ, dabere na ihe mgbaàmà.
Iji cupping stenokardicheskie agha n'ihu ndị na-abịa anụ ahụ ma ọ bụ nrụgide mmetụta uche ndị pụrụ ime ka nnukwu, na-egbu oge respiration, na ọrịa na-enweta site 1 3 doses na etiti oge nke 30 sekọnd n'etiti injections. Dịkwuo onunu ogwu enweghị elekọta ọkachamara amachibidoro.
Na ikpe nke-enyo enyo na exacerbation nke obi bara ma ọ bụ myocardial infarction, nnukwu n'elu ndidi na-enweta site 1 3 doses n'okpuru ike akara nke ma obi ọnụego na ọbara mgbali. Ọ bụrụ na ọ dịghị mma, mgbe ahụ, usoro a ugboro ugboro nkeji ise gasịrị site a na mkpebi nke dọkịta. Na ọzọ nkeji iri, ọnọdụ ga-akawanye. Ma ọ bụghị ya, ị nwere ike ikwugharị mkpachapụ ọzọ n'okpuru nlekọta nke a dibịa.
Tupu ọgwụgwọ usoro cupping akwara spasm (n'ihi na-achọpụta ọrịa ma ọ bụ ọgwụgwọ catheterization) ndinọ onye ọrịa site injection 1-2. Mgbe e nwere mkpa onunu ogwu nwere ike ugboro ugboro, ma ọ bụrụ na akara kwa ọbara ekesa.
Specific nwere ikwu maka ojiji nke a ịgba
N'ọnọdụ mgbe a ọhụrụ ịgba na-etinyere maka oge mbụ, ma ọ bụ mgbe ikpeazụ dose kemgbe ihe karịrị awa 24, ọ bụ ihe amamihe na-eduzi mbụ pịa na ikuku, n'ihi na ọ na-apụghị ichedo chọrọ onunu ogwu. N'ihi na doses dị na ntụziaka nebulizer nọgidere enwe ọgwụgwụ, na mgbe ahụ wepụtara. N'oge ojiji na a ịgba karama dispenser ga-upwardly na ekwesị.
Nyocha ọkachamara na-egosi na elu onunu ogwu nke ọgwụ, ọ bụ mgbe ahụ ma ọ bụ n'oge Ịhazi ojiji pụrụ iduga ndidi mmepe na ndidi. Ndị dị otú ahụ a atụmatụ na-mepụtara na ojiji nke ọgwụ ọjọọ ndị ọzọ na-ekewet nke nitrati. N'ọnọdụ dị otú ahụ, ndị dọkịta nwere ike ikwu iji kagbuo ojiji nke ọgwụ maka 2-3 ụbọchị, mgbe a N'ezie nke mgbe omume, nke e kere 3-6 izu, na-ezumike maka 3-5 ụbọchị, na-eji dochie ya na nwa oge site ọgwụ ọjọọ ndị ọzọ na yiri mmetụta. N'ọnọdụ ka ukwuu, mgbe otu nkwụsị ma ọ bụ discontinuation uche nke onye ọrịa kama ngwa ngwa weghachiri eweghachi. pụtara mmiri ewepụtara metabolites dị ka akụrụ fọrọ nke nta zuru.
Ọnụọgụ ọgwụ na ngwa ngwọta
Dị ka chọrọ na ntụziaka nkwadebe "Izoket" (maka infusion ngwọta) etinyere intravenously. The onunu ogwu nke n'imeso vrechom n'otu n'otu ahaziri iji hemodynamic na-adakarị kwa nke onye ọrịa. Agwọ ga-amalite na a ala dose ma na-amụba nwayọọ nwayọọ eme ka chọrọ ego. Ntuziaka na-atụ aro usoro onunu ogwu bụ 2-7 mg / Ọrụ Nchịkwa, karị, nkezi dose bụ banyere 7.5 mg / Ọrụ Nchịkwa. N'ọnọdụ nke oké mkpa olu nwere ike mụbara ka 10 mg / Ọrụ Nchịkwa.
N'ọnọdụ ka ukwuu, ndị mmadụ na obi odida achọ elu doses nke ọgwụ. The mmeghe nke ọgwụ kwesịrị ịbịa inpatient ọgwụgwọ n'okpuru nlekọta nke a ọkachamara na ojiji nke akpaka usoro maka infusion. The dum usoro na-esonyere akara egosi mgbasa (ọbara mgbali na obi ọnụego).
- ka a ịta nke 0.01% (100 micrograms / ml) - 50 ml nke 0,1% ọgwụ nwere ike ime ka 500 ml nke nkwadebe njikere maka ochichi;
- ka a ịta nke 0,02% (200 micrograms / ml) - 100 ml nke 0,1% ngwọta nke ọgwụ nwere ike 500 ml nke agwọ ọrịa njikere maka ochichi.
Contraindications na-elezi anya na
The ọgwụ na-adịghị gosiri maka ọrịa hypersensitive ka nitrate ogige, dị ka nke ọma dị ka ndị ọzọ na ihe nke aerosol "Izoket". The ngwa na-egbu ma ọ bụrụ na ọrịa dị otú ahụ ọrịa:
- hypotonia, na nke systolic mgbali bụ n'okpuru 90 mm HG.;
- vaskụla insufficiency na nnukwu ogbo, e.g., n'oge ujo ma ọ bụ vaskụla ida;
- pericarditis na pericardial tamponade;
- na cardiogenic ujo ikpe ebe e nweghị ekwe omume na-agbanwe ndị ọzọ ụzọ mgbali na ekpe ventricle nke obi;
- hypertrophic cardiomyopathy;
- mmechi glaucoma.
Ke adianade do, ọgwụ na-adịghị gosiri n'ihi ndị na-n'okpuru iri na asatọ afọ. Ntuziaka maka ojiji na-atụ aro na ojiji nke ọgwụ ọjọọ na oké ịkpachara anya na n'okpuru elekọta ya mgbe nile dị otú ahụ ikpe:
- myocardial infarction na nnukwu eruba mgbe onye ọrịa nke a belatara mgbali ekpe obi ventricle ndochi;
- ụba intracranial mgbali;
- mitral na / ma ọ bụ aortic stenosis;
- ịchọputa omume puru onye ọrịa orthostatic ọrịa na ụkpụrụ ọbara ekesa;
- gbasara akụrụ ma ọ bụ mmebi imeju.
Pregnancy na lactation
Ọkà mmụta sayensị na mmepe nke ọgwụ anụmanụ ọmụmụ e duziri. The nnwale na ule gosiri na mmetụta na-ebibi na nwa ebu n'afọ na-adịghị rụrụ.
Mmekọrịta ndị ọzọ ọgwụ ọjọọ eme ihe
A machibidoro iwu ịkọrọ vasodilators na "Izoket" nkwadebe (ịgba). Ha were na Nchikota nwere ike ime ka ụba hypotensive mmetụta. Otu mmetụta gụnyere imekotaotuugbo n'ikuku "Izoket" na ndị dị otú ahụ aerosol ọgwụ: antihypertensives, calcium ọwa blockers, "Quinidine" ma ọ bụ "novokainamid" neuroleptics, 5-phosphodiesterase inhibitors.
Esiwanye ike antianginal mmetụta mgbe eji na njikọ na ọgwụ ọjọọ ndị dị ka "Amiodarone", "propranolol", "Nifedipine", "Verapamil," na ndị ọzọ na blockers nke calcium ngwa ngwa ọwa.
Mụbara intracranial mgbali na a ọrịa nwere ike ime n'oge Nchikota ọgwụ na atropine na ndị ọzọ na m-holinoblokatorami.
Oké ọnụ ke ọbara mgbali, na-eduga akwara perfusion, na-egosi n'okpuru nduzi nke Alfa-blockers na sympathomimetic.
Mmetụta na reviews
Ntuziaka kọwara na a ọtụtụ mmetụta na e nwere ike mere site na ọgwụ ọjọọ, "Izoket" (ịgba). Nyocha nke ụfọdụ ndị ọrịa emeso ya na a ọgwụ, na-egosi na ọdịdị nke isi ọwụwa, nke na nkà mmụta ọgwụ na-akpọ "na nitrati". Dị ka a na-achị, mgbe 2-3 ụbọchị nsogbu kpamkpam na ya na-adịghị achọ ka mgbazi. Kama ịdị agwọ ọrịa nwere ike ime ka phenomena dị ka ọgbụgbọ, nācha ọbara-ọbara nke anụ ahụ, vomiting, na akọrọ ọnụ.
Otú ọ dị, dị ka reviews, ọrịa na-achọpụta na nrụpụta ọrụ. Na mgbe na-anata na dị na ọkachamara chọrọ nke mmetụta na-adịghị ime otú ahụ ugboro ugboro. Ewezụga bụ ndị isi na-awa n'ụbọchị ndị mbụ nke iji, nke so ọtụtụ nke ikpe, ma na-emekarị na-aga ụbọchị ole na ole.
Uku karịa olu
An ovadozu nke ọgwụ nwere ike ime ka a ọnụ ọgụgụ nke oké njọ deviations: syncope, ida, elu intracranial nsogbu, hyperthermia, ọdụdọ, visual ọrụ ọrịa, ubara sweating, methemoglobinemia, bradycardia, mkpọnwụ, na amaghị onwe ya. Ọ bụ ya mere ọ dị mkpa na-onwe-obi, ma na-ọgwụ nditịm dị ka chọrọ nke a ọkachamara!
Ọ bụrụ na ihe mgbaàmà kọwara na-achọ mwepụ nke ọgwụ na-eduzi ọgwụ iji na kwụsie ike ọrịa na-arịa.
analogs
Agwọ ọrịa "Kardiket» (CHWARZ PHARMA, Germany) - otu n'ime ndị kasị ọnyà ọgwụ ọjọọ (analogs) nke ọgwụ "Izoket" (ịgba). The price nke a dochie anya bụ dabere na ịta nke nọ n'ọrụ umi na ọnụ ọgụgụ nke mkpụrụ ọgwụ na a ngwugwu.
Ka ihe atụ, gị n'ụlọnga ke mbadamba 20 mg "Kardiket ghara" (20 PC. On ngwugwu) bụ site 62 72 rubles, mgbe otu nkwadebe, naanị na a onunu ogwu nke 40 mg mbadamba na nke ukwu nke 50 iberibe, nwere a uru nke 210-220 rubles.
A ìgwè nke ọgwụ "Nitrosorbid" arụpụtara site ọtụtụ Russian ụlọ ọrụ, na-enwe ụdị dị iche iche nke tọhapụ, kwa, bụ a dochie anya ọgwụ "Izoket". Analogues nke otu a nwere aha "Nitrosorbide-Rusfar", "Nitrosorbide", "Nitrosorbide NS", "Nitrosorbide-UWI."
eri nke
Na Russian pharmacies ga-akwụ site na 365 na 470 rubles kwa onunu ogwu Nwa "Izoket" (ịgba). The price na-kpụrụ dabere na ọnọdụ nke retail tinyekwa na ya ọnọdụ. Na weebụsaịtị na-ere ọgwụ ike zụrụ na a ala na-eri karịa a ot ahịa ọgwụ nso n'ụlọ gị. Ma mgbe ịtụ n'elu Internet ga-akwụ 200 rubles maka nnyefe ma ọ bụ na-enweta a free gị n'ụlọnga na paragraf ex, nke a na ọ bụghị mgbe niile conveniently odude n'ọdịdị ya.
Ọzọkwa, n'oge ọ bụla na-ere ọgwụ ị nwere ike ịzụta ngwugwu (10 vials) lekwasị ngwọta maka infusion "Izoket". Ya price dịgasị si 906-980 rubles.
Isi
The ọgwụ na-arụpụtara site German ụlọ ọrụ "YUSB Pharma GmbH". Adị ndụ nke afọ ise. Okwu nke ire - ọnụnọ nke a dọkịta ọgwụ. Mgbe ogologo oge nke iji ya na-atụ aro iji chọpụta arụmọrụ nke sprayer. Labelụ nke aerosol na-adọrọ mmasị na ala akụ. Mgbe mmiri mmiri rute n'ogo ọ kwesịrị ka a ọgwụ ọhụrụ, ebe ọ bụ ojiji nke otu dị na karama bụ nanị kwe omume na a obere weturu, nke na-aṅụ ara tube na-mikpuru na mmiri mmiri.
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