Ahụ ike, Preparations
Mikoflyukan: ntuziaka maka ojiji
onunu ogwu ụdị
Nkwadebe "Mikoflyukan" ntụziaka maka nke a na-egosi n'okpuru ike-emepụta n'ụdị mbadamba na dị iche iche kasịnụ nke nọ n'ọrụ umi ma ọ bụ n'ụdị ihe ngwọta maka infusion. The mbadamba na-acha ọcha, gburugburu udi na ubé bevelled n'ọnụ ya.
Na mbadamba nwere 50 mg nke nọ n'ọrụ umi na ma akụkụ nke echiche «F», na ndị ọzọ - "50". The mbadamba ụdị "Mikoflyukan" 150 mg nke nọ n'ọrụ mgwa - «F150» na n'ikewa akara, karị.
The ngwọta nkwadebe bụ colorless, uzo, na-enweghị ihe ọ bụla ahụ.
Mejupụtara: Mbadamba
Active umi: fluconazole - 50/150 mg (1 tab.).
Excipients:
- sịlịkọn dioxide ,
- lactose,
- povidone,
- magnesium stearate
- Valium,
- talc,
- cellulose mikrokristallicheskayae
ngwọta
Active umi: fluconazole - 2/200 mg (1 ml mkpọ na 1, karị).
Excipients:
- Mmiri maka ịgba ntụtụ,
- sodium chloride.
The pharmacological edinam nke ọgwụ "Mikoflyukan"
Guide na-ekwu na nkwadebe akọ antifungal mmadụ nke triazole emepụta. Fluconazole inhibit ergosterol njikọ dị ka ndị a: ọ na-enye ndị permeability nke na cell mgbidi. The ọgwụ na-arụ ọrụ megide Microsporum, Candida, Trichophyton, Cryptococcus neoformans.
A atụmatụ nke pharmacological edinam nke ọgwụ bụ na ọ bụ ma nhọrọ inhibitor nke cytochrome P450 na fungi, ma n'otu oge, adịghị egosi na ihe ọ bụla ọrụ megide a enzyme usoro mmadụ.
Pharmacokinetics
The ọgwụ na-ọma-etinye obi gị dum mgbe ochichi, na nri oriri na njikọ na-ewere ọgwụ adịghị emetụta ya absorption. Bioavailability - 90%. The ọgwụ na-ekesa nile akụkụ na anụ ahụ nke ahụ. N'ihi ya ya ịta na plasma ịta hà na-esonụ akụkụ na anụ ahụ: nkwonkwo ọmụmụ, mmiri ara, asu, mmamiri secretions, sputum na perinatal ọmụmụ, na cerebrospinal ọmụmụ bioavailability nwere ike mbio 50 90%.
Ọzọkwa, ụfọdụ akụkụ na anụ ahụ nke ọgwụ ịta ike gafere ịta na plasma. N'etiti ha, ndị epidermis, na dermis, na stratum corneum, ọsụsọ mmiri mmiri. The ọkara ndụ - banyere 30 awa.
Egosi maka ojiji nke ọgwụ "Mikoflyukan"
Iwu ahụ kwuru na ọgwụ nwere nnukwu ọrụ megide microorganisms ndị na-esonụ ọrịa, nke na-ewekarị fungal-efe efe:
systemic candidiasis,
cryptococcosis,
mucosal candidiasis,
mmamiri candidiasis,
mgbochi nke fungal-efe efe
akpụkpọ mycoses,
onychomycosis,
pityriasis versicolor,
parakoktsidiovikoz,
coccidioidomycosis,
pistoplazmyuoz,
sporotrichosis.
Mmetụta nke ọgwụ "Mikoflyukan"
Nyocha nke ule otu mgbe a na usoro nke ọmụmụ nke ọgwụ, gụnyere placebo-ule na ụzọ ndị ọzọ nke nnyocha gosiri na ọgwụ ike ndị na-esonụ mmetụta:
- na ùgwù nke digestive tract:
abdominal mgbu,
ọgbụgbọ,
flatulence,
afọ ọsịsa;
- na ùgwù nke Central ụjọ usoro akụkụ:
dizziness,
isi ọwụwa;
- banyere nfụkasị Jeremaya:
anaphylactic Jeremaya mere nke organism,
akpụkpọ ọkụ ọkụ.
Contraindications ọgwụ "Mikoflyukan"
Ntuziaka ka ọgwụ na-ekwu na ndị contraindications ya n'ikuku bụ obere ezu, n'etiti ha:
ruo 1 afọ,
afọ ime,
uche na triazole compound na fluconazole.
ọgwụ interactions
Prothrombin oge na-abawanye mgbe ojiji nke ọgwụ ọjọọ anticoagulant coumarin ụdị.
Nkwekọrịta nke sulfonylurea onu hypoglycemic mmadụ budata dịkwuo ha ọkara ndụ na kọntaktị na fluconazole.
Fluconazole ọkara ndụ oge na-ebelata mgbe kpọtụụrụ na rifampicin.
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