Ahụ ikePreparations

"Mydocalm": ihe na-enyere, nkọwa nke ọgwụ, contraindications

Gịnị bụ a ọgwụ ọjọọ, "Mydocalm"? On ihe na-eme ka ngwá ọrụ a? Egosi na atụmatụ nke a ọgwụ, anyị na-ewetara n'okpuru. Ị ga-amụtakwa banyere otú na-emeso a ọgwụ, ole ọ na-efu na ihe ọ nwere.

Ụdị nke ọgwụ ntọhapụ, nkwakọ, nkọwa, mejupụtara

Na ihe ụdị ahịa ọgwụ ọgwụ ọjọọ, "Mydocalm" abịarute (site na ihe na-enyere nke a na nkà mmụta ọgwụ, anyị na-akọwa n'okpuru)? The ngwá ọrụ dị na mbadamba na-na a ngwọta zubere maka parenteral ochichi.

Gburugburu na-acha ọcha "Mydocalm" mbadamba, na price nke na-egosi n'okpuru, mejupụtara tolperisone hydrochloride. Dị ka n'ihu Efrata nke ọgwụ na-atụle: anhydrous colloidal silicone, citric acid monohydrate, ọka starch, stearin, hydroxypropylmethyl cellulose 2910, talc, Macrogol 6000, microcrystalline cellulose, colorant, lactose monohydrate na titanium dioxide.

Dị na ọnya Ukwu bụ ụzọ, nke na-enịm ke igbe mere nke akwụkwọ.

The putara ihe "Mydocalm" na ampoules nwekwara tolperisone hydrochloride na lidocaine. Ke adianade do, ọgwụ na-agụnye ndị na-esonụ Efrata: talc, citric acid monohydrate, lactose monohydrate, silicone colloidal anhydrous, macrogol 6000, microcrystalline cellulose, stearin, titanium dioxide, ọka starch, nwa ígwè oxide, hydroxypropylmethyl cellulose 2910, ígwè oxide uhie odo ígwè oxide.

Drug "Mydocalm" na ampoules dị na plastic containers, nke na-enịm ke igbe mere nke kaadiboodu.

Key Njirimara

Gịnị bụ a "Mydocalm"? On ihe na-eme ka a ọgwụ? Dị ka ntụziaka, isiokwu gị n'ụlọnga na-ezo aka muscle relaxants aminoketonovoy otu nke nwere a Central mmetụta.

The nrụpụta ọrụ nke a ọgwụ a na-ejikọta ya na ụkpụrụ nke na-arụ ọrụ ibe (caudal) nke reticular guzobere. Iji nke agwọ ọrịa na-akwalite mgbochi nke mụbara excitability nke ọkpụkpụ azụ mpiaji. Ọ na-emetụta akwara (elu).

atụmatụ ọgwụ

Nkwadebe "Mydocalm" (ndakọrịta nke ngwá ọrụ na ndị ọzọ na-anabata, ma n'okpuru kpọmkwem ọnọdụ) bụ H-anticholinergic. Ya nọ n'ọrụ gị n'ụlọnga nwere a-eguzosi ike na akpụkpọ ahụ nke bụ isi akwara (afferent), na motoneurons. Nke a pụrụ isi kwuo ya bụ n'ihi na ọgwụ ya ikike inwe mmetụta n'ahụ ọrụ nke mpiaji spinal synapses.

Ọzọkwa mara na nke a ọgwụ ọjọọ a abụọ oge slows ala neurotransmitters. Na nke a emee ruru ka mgbochi nke calcium ntinye usoro na synaptic Ọdịdị, nke na-emi odude ke akwara ozi.

Mmetụta nke ọgwụ na reticulospinal ụzọ karịsịa akpọ mgbe decelerating excitation Filiks. N'otu aka ahụ mestnoanesteziryuschee achọpụtara na edinam nke ọgwụ (n'ihi na ọdịnaya nke lidocaine nime ya).

The kinetics nke ọgwụ

Atụle gị n'ụlọnga na-ọma etinye obi gị dum na gootu. Ya ịta (max) a ruru mgbe 65 nkeji mgbe na-ewere ọbara. Drug metabolism pụtara na imeju na-na akụrụ. Tolperisone nkwekọrịta ịpụta na mmamịrị.

Ugboro ugboro N'ezie "Mydocalm" enweghị mmetụta na akụrụ na imeju na, nakwa dị ka usoro nke hematopoiesis.

The ngwá ọrụ mbelata rigidity na experimentally rata muscle hypertonicity. Ọgwụ Njirimara nke ọgwụ na-eji ọtụtụ iji belata muscle erughị ala na-enweghị nchịkwa na hypertonus na na-metụtara extrapyramidal ọrịa.

Ọ kwesịkwara kwuru na ọgwụ na-akwalite ọrụ nke onye (ya mmegharị). Ke adianade do, o nweghị mmetụta na-arịa ọrịa cortex, n'ụzọ zuru ezu na-echebekwa ndị ọrịa larịị nke wakefulness.

Dị ka ntụziaka, ọgwụgwọ "Mydocalm" Akpọlite ubé akpọ antispasmodic na adrenoceptor igbochi mmetụta. N'ihi nke a, ọ ka mma anụ ahụ perfusion.

Ke N'ezie nke ogologo oge na-adakarị ọnwụnwa nke a gị n'ụlọnga nwere a akpọ mmetụta na ọbara na akụrụ ya.

Drug "Mydocalm": ihe na-enyere?

The ngwá ọrụ gosiri maka ojiji na ndị na-esonụ mgbe:

  • Na ụmụaka na-eme, na ihe mgbaru ọsọ nke ọgwụ Little ọrịa (ie, spastic mkpọnwụ). Ke adianade do, a ọgwụ na-eji na a dị iche iche si malite encephalopathy na mgbaàmà nke muscle dystonias.
  • N'okpuru ọnọdụ ndị na-na-ebu a enweghị nchịkwa hypertonus nke striated muscle anụ ahụ ruru ndị na-emepe emepe pathologies (akwara ozi) organic (e.g., multiple sclerosis, encephalomyelitis, myelopathy, mmapụta mmetụta nke ọrịa strok, pyramidal tract ọnya).
  • N'okpuru ọnọdụ nke ịmaliteworị dị ka a n'ihi nke mmebi vaskụla innervation (e.g., acrocyanosis, angioneurotic disbazii intermittent uwa).
  • Mgbe muscular hypertonicity, contracture nke uru ahụ na-eso ọrịa nke akụkụ nke ije (eg, spondylosis, ogbu na nkwonkwo nke n'ikpere aka, na ikpere na nkwonkwo úkwù, spondylarthritis, ọrịamkpokọta nke lumbar na cervical).
  • Mgbe post-thrombotic venous ọbara ọrịa na lymphodynamics.
  • Dị ka mbenata postoperative ọgwụgwọ na orthopedic na trauma omume.
  • Mgbe trophic onya kpụrụ na ala na nsọtụ, angiopathy (gụnyere diabetogenic), thromboangiitis obliterans angiosclerosis na, nakwa dị ka autoimmune ọrịa na (Raynaud ọrịa na systemic sclerosis).

Bans ojiji

Mgbe ụfọdụ, i nwere ike na-ekenye a Erere, injectables "Mydocalm"? The ojiji nke a ọgwụ na-contraindicated na:

  • myasthenia gravis;
  • hypersensitivity ka tolperisone na mara allergies ka lidocaine;
  • n'okpuru afọ atọ na ọnwa (na mbadamba ụdị otu afọ).

dosing

Atụmatụ nke ngwá ọrụ e debere dọkịta dabere na ọrịa, na ọgwụ ọjọọ tolerability.

N'ihi na okenye na ụmụ mmadụ agwọ ọrịa na-ndinọ ke ichekwa 150-450 mg (kwa ụbọchị dose) na atọ nzọụkwụ. The malite onunu ogwu nke a ọgwụ bụ 50 mg ugboro atọ n'ụbọchị. Na enweghị irè nke ya na-abawanye.

N'ihi na intramuscular ogwu ogbugba, ọgwụ na-eji na ego nke 200 mg kwa ụbọchị (abụọ ọgwụ) na igba ogwu n'akwara - 100 mg (otu ugboro kwa ụbọchị). Nke abụọ ahụ ọ na-achọ a nnọọ ngwa ngwa infusion nke ọgwụ.

Maka ụmụaka okenye karịa ọnwa atọ (ruo 6 afọ) na onunu ogwu nke ọgwụ n'okpuru echiche na gbakọọ dị ka ndị a: 5,10 mg kwa n'arọ ahu arọ (ugboro atọ kwa ụbọchị). N'ihi na a na nwa 7-14 afọ na-atụ aro iji a mbadamba na a kwa ụbọchị dose nke 2-4 mg kwa n'arọ nke ahu (ugboro atọ kwa ụbọchị).

Oral nlekọta "Mydocalm" ga-achọkwa na nri.

edinam n'akụkụ

Na-ewere ọgwụ na onye hypersensitivity nwere ike ime ka ike na uru, dyspeptic phenomena nke ọdịdị (ọgbụgbọ, ahụ erughị ala na vomiting) na isi ọwụwa.

Na ngwa ngwa igba ogwu n'akwara infusion ngwọta nwere ike ibelata ọbara mgbali.

Ọ bụrụ na ị na-hypersensitive ọgwụ ịzụlite nfụkasị Jeremaya. Dị ka a na-achị, nta doses ọgwụ mmetụta bụ nnọọ ngwa ngwa.

ọgwụ interactions

Ozi banyere mmekọrịta, nke egbochi ndị ngwa nke ngwaahịa a na-adịghị. Otú ọ dị, ọ ga-ahụ kwuru tolperisone na-enwe mmetụta Central ụjọ usoro. N'ihi ya ọgwụ adịghị eme ka iro ụra, n'ihi ya, ọ nwere ike ikpokọta na hypnotic na ogwuura, nakwa dị ka ọgwụgwọ nwere a ethanol.

Mgbe imekotaotuugbo nlekọta "Mydocalm" niflumic acid enhances mmetụta. Ọ bụrụ na ọ dị mkpa, a Nchikota dị otú ahụ mmadụ nwere ike ịchọ dose Mbelata nke ikpeazụ.

Elu muscle relaxants, ọgwụ ọjọọ maka general ná Nkụnwụ na psychotropic bekee, dị ka nke ọma dị ka "clonidine" welie irè nke tolperisone.

Na-eri na reviews

Ole bụ "Mydocalm"? The price nke a gị n'ụlọnga bụ banyere 185 rubles.

Nleba ikweta na ọgwụ na ajụjụ na-egosipụta onwe ukwuu n'ụzọ dị irè, karịsịa na ọrịa nke nkwonkwo. Ke adianade do, ngwá ọrụ a dị nnọọ mma maka ọbara na ụbụrụ, gụnyere bilitere mgbe traumatic mmerụ ahụ n'ụbụrụ.

Otu n'ime ihe ndị na-ezighị ezi reviews nwere ike mata site ndị na-ekwu na ndị ọgwụ ọjọọ, "Mydocalm" bụghị a panacea. Ọtụtụ mgbe, nke a ọgwụ na-eji dị ka a na-arụzi ọgwụgwọ.

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