Ahụ ike, Preparations
Ngwa ntụziaka, nzaghachi na analogue "Locri"
Hypertensive ọrịa obi na ọrịa bụ nnọọ nkịtị na ụwa. Nke a bụ a pụtara ogbu na nwayọọ ọrịa, nke bụ ná mmalite nkebi bụ ike ịmata. N'ihi ya, mgbe afọ 40, ha kwesịrị ịna-nyochaa arụmọrụ dvleniya. Ọ bụrụ na-arụpụta bụ oke elu, ị kwesịrị ị na ịkpọtụrụ dọkịta gị. The mbụ ọgwụgwọ amalite, ndị ngwa ngwa i nwere ike imeri ọrịa ahụ.
Modern ọgwụ ọjọọ na-ji elu arụmọrụ. Otu a nke blockers. Mbadamba nnọọ nwayọọ belata ọbara mgbali na adịghị imerụ ahụ. Nnọọ na-ewu ewu n'etiti ndị na-agwọ ọrịa taa bụ na nkwadebe "Lokren". Ntuziaka maka ojiji, analogs, na ezi usoro onunu ogwu - a nile a otú n'okpuru.
The mejupụtara nakwa ụdị ọgwụ ntọhapụ
Mbadamba "Lokren" na-acha ọcha, ubé convex na otu akụkụ na-akara na e dere EK20. Dị otú ahụ na a titer nke na nkà mmụta ọgwụ nwere ike n'ụzọ dị mfe na-akwanyere ùgwù si nwere. The mbadamba na-kpuchie na a mkpa shei. The isi akụrụngwa na mejupụtara nke mbadamba nkume a na-ewere gidrohrorid betaxolol 20 mg. Auxiliaries ọgwụ ndị lactose monohydrate, microscopic cellulose, sodium karboksilmetilkrahmal.
Shei na-emi esịnede gipromilozu, macrogol, titanium dioxide. Dị na mbadamba a ọnya, na 14 iberibe na onye ọ bụla. Ọ bụla analogue "Locri" ga-enwe a yiri mejupụtara na-egosi maka ojiji.
Mmetụta nke ọgwụ na ozu
Mbadamba nke a ìgwè nke beta-blockers. Ha na-ahuta ka nhọrọ blockers nke mbụ n'usoro. Betaxolol, nke bụ akụkụ nke ọgwụ, nwere cardioselective beta-adrenoceptor igbochi mmetụta, ji enweghị agonist ọrụ bụ na-adịghị ike akpụkpọ ahụ. N'ihi nke a na ọgwụ ọjọọ na-ebelata obi ọnụego n'oge ezumike na emega ahụ. The isi mmetụta - ebelata ọbara mgbali na-ezu ike na n'oge omumu.
Mgbe na-eji ọgwụ na-aga tachycardia, belata ibu na obi, nkịtị elu ọbara ekesa. Antihypertensive mmetụta nke betaxolol na ruo ogologo oge iwere na-adịghị belata. Mgbe otu ingestion dose mbadamba nkume ndị ahụ ọgwụgwọ mmetụta emee n'ime awa atọ na-aga n'ihu ofụri usen. Anụ pụta ga-enweta na clusive ọgwụgwọ. Ndị dị otú ahụ nwere na ozu mkpụrụ ọgwụ "Lokren". Drug analogues nwekwara apụta ọbara egosi mgbe eji n'ụzọ ziri ezi.
Pharmacokinetics
Mgbe ingested, ọgwụ ngwa ngwa dissolves na bụ 100% etinye obi gị dum na afo. The kacha mmetụta na-enweta mgbe abụọ awa plasma. The ọgwụ na-ejikọ na ọbara esenyịn site 50%. Betaxolol na imeju Nleta ihe-adịghị ejekwa ozi metabolites. Fọrọ nke nta 80% nke nọ n'ọrụ mgwa anyụpụ site akụrụ n'ụdị metabolites. 20% na-abịa site ahụ agbanwebeghị.
Ngwa ngwa-ekwe omume inwe a mma ọgwụgwọ mmetụta, ma ọ bụrụ na kwesịrị ekwesị iri mkpụrụ ọgwụ "Lokren". Ntuziaka maka ojiji nwere niile ozi ndị dị mkpa.
Egosi na contraindications
Ihe kpatara nke nhọpụta nke ọgwụ a na-ewere ọbara mgbali. N'aka e nwere ike iwere naanị ma ọ bụ na Nchikota na ọgwụ ndị ọzọ iji belata nsogbu. Mbadamba e kenyere iji gbochie ọrịa strok na.
Contraindications ọgwụ ọgwụgwọ a na-ewere oké bronchial ụkwara ume ọkụ na-adịghị ala ala bronchitis, nnukwu obi ọdịda. Ejila ọgwụ na owụt phenomena bradycardia, oké iche nke Raynaud ọrịa na elu ọbara nsogbu. E nwere afọ ókè. Ọgwụ adịghị kenyere obere ọrịa.
Ọ na-adịghị atụ aro na-aṅụ mbadamba ọrịa na gbasara akụrụ ma ọ bụ hepatic insufficiency. N'oge ime na lactation ngwá ọrụ ike ga-eji naanị ma ọ bụrụ na ndị nwere uru nne kari ike imerụ nwa ọhụrụ.
Tupu ọgwụgwọ ga-akpachara anya na-agụ ntụziaka na nke ego "Lokren". Ọbịa ọkachamara na-atụ aro na mmetụta na-erukwa na ndị ọrịa na-adịghị rube isi na-atụ aro.
onunu ogwu
The ọgwụ kwesịrị iwere na ọtụtụ mmiri. The na nkà mmụta ọgwụ na-ekwesịghị-ata ata. Ọgwụgwọ ga-amalite na a ọkara mbadamba (10 mg). Ọ bụrụ na a mma ọgwụgwọ mmetụta, ọ dị mkpa ka iwelie onunu ogwu adịghị abịa izu abụọ. Oke kwa ụbọchị ọnụego nwere ike gafere 40 mg.
Ọtụtụ ndị dọkịta adịghị ike ikwu na ha na-agwọ na-aṅụ ihe karịrị otu Erere kwa ụbọchị. Ọ bụrụ na ị nwere ogbenye mgbali Mbelata dị mkpa iji tinye ọzọ antihypertensive ọgwụ ọgwụgwọ. Ọrịa na oké gbasara akụrụ insufficiency ga amalite na-ewere ọgwụ na a dose of 5 mg. Nke nta nke nta dịkwuo ọnụego ya kwa ụbọchị. Ọ nwere ga-amụ tupu eji n'aka "Lokren" ntụziaka ntuziaka.
ovadozu
Na ihe ovadozu ọgwụ nwere ike vertigo, elu nsogbu dobe, cyanosis nke mkpịsị aka na mbọ, bradycardia, lightheadedness. Ọzọkwa ịzụlite mgbaàmà ndị dị otú ahụ dị ka bronchospasm na obi ọdịda.
Ọgwụgwọ nke ovadozu mejupụtara gastric lavage. Ọ na-atụ aro ka na-aṅụ a ndidi adsorbent na ejikọrọ infusion ọgwụ. Nnọọ ọnụ ke mgbali dị mkpa prokapat "dopamine" na-abanye "Atropine". Ị ga-hoo haa tinye gbasara obi glycosides na antispasmodics. Na oké ikpe, ọ na-egosi iwebata ọbara nọ n'ọnọdụ na plasma. Ọ bụla analogue "Locri" ga-, na-esonụ na onunu ogwu kenyere site dọkịta.
mmetụta
Mgbe n'imeso ọgwụ anabata nwere ike amalite. Ọ na-egosipụta onwe ya n'ụdị a ọkụ ọkụ na akpụkpọ itching. Ọzọkwa, e nwere ndị Jeremaya mere na akụkụ nke ụjọ usoro, nke na-egosipụta site dizziness, isi ọwụwa, asthenia, ehighi ura, na-arọ nrọ, paresthesia. Mmetụta na-agụnye ebelata ọhụụ, na ibelata intracranial nsogbu. Na oge nke na-ewere ọgwụ na-emekarị hụrụ abdominal mgbu, ọgbụgbọ, vomiting. Nwere ike ịgbanwe ọbara na ịzụlite leukopenia. Men na-ewere ọgwụ na-akpatakarị enweghi ike. The ịkpachara anya ga-họpụtara ọgwụ na agadi.
Ọ ga-echekwara na ụlọ okpomọkụ n'ebe gbara ọchịchịrị keerughi ụmụ, ọgwụ "Lokren". Analogs mee ihe n'otu ọnọdụ.
Analogue "Locri" na Russia - ọgwụ "Betaxolol"
Olee otú ịhọrọ a quality dochie anya ọgwụ? Gịnị ma ọ bụrụ na ndị ahịa ọgwụ enweghị pụtara "Lokren"? Drug analogues ga mgbe nile na-enwe ike nwere ike ikwu na a dọkịta. Popular n'aka "Betaxolol." Ọ cardioselective beta-blocker eji belata ọbara mgbali na rịaworo ọgụ. Mgbe ingestion kpamkpam rapara ke afo. The kacha mmetụta na-enweta na a plasma awa atọ. The ọgwụ anyụpụ site akụrụ n'ụdị metabolites na-guzobere na imeju.
The ọgwụ lowers intraocular mgbali nke ọma, ma ọ bụrụ na ị na-eji ihe ngwọta na ụdị anya tụlee.
The na nkà mmụta ọgwụ na-eji otu ụbọchị na a onunu ogwu nke 20 mg. Ọgwụ nwere ike iwere naanị ma ọ bụ dị ka akụkụ nke Nchikota ọgwụ. Ọ bụghị na-atụ aro maka ojiji n'oge ime na lactation. Na obere okwu, ndị ọgwụ ọjọọ na-akpata mmetụta n'ụdị a ọkụ ọkụ na a na-ere sensashion na akpụkpọ. Ọzọkwa, e nwere ike ịbụ dizziness na ọgbụgbọ, nakwa dị ka eji mbadamba nkume "Lokren". Russian analogues nwere otu na-egosi na contraindications.
Drug "Betacam"
Ọgwụ bụ beta-blocker ariri mbu. ọcha ọgwụ. Onye ọ bụla dose ẹdude 20 mg nke betaxolol hydrochloride. Ọgwụ nwere ike kenyere naanị site dọkịta. The ọgwụ na-enyere aka normalize ọbara mgbali, belata obi ọnụego na-ezu ike na n'oge omumu, ọ na-eduga nkịtị elu ọbara na aka rịaworo.
Ọ bụghị na-atụ aro maka nkà mmụta ọgwụ na pathologies nke akụrụ na imeju. N'oge ime na lactation ọgwụ ajuru aju. Ukwu nwere ike ime ka nfụkasị Jeremaya mere na nta deviations na ụjọ na digestive usoro. Kwesịrị ịkpachara anya maka kenyere ndị agadi na na ikpe nke na hypersensitivity na mmiri nke na mbadamba. Nke a analogue "Locri" ike kpamkpam dochie dị mbụ.
Nyocha
About Beta-blockers ọkachamara-ekwu okwu ọma. N'ihi na a obere oge ọ bụ ike normalize na kwa nke nsogbu na belata ekpe ventricular hypertrophy. Ọgwụ ndị a na-ọma na-anabata na-adịghị emetụta ọrụ ndị ọzọ na akụkụ na usoro. Ọ bụla analogue "Locri" ga-egosi mmetụta dị mma ma ọ bụrụ na ọ na-eji dị na ntụziaka.
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