Ahụ ike, Preparations
"Fliksotid": ntuziaka maka ojiji, reviews. ọgwụ analogues
Ị maara ihe ọgwụ "Fliksotid" pụtara? Ntuziaka maka ojiji nke ọgwụ, ya na-egosi, mejupụtara, mmetụta na ntọhapụ ụdị ga-kọwara n'ụzọ zuru ezu n'okpuru. Ke adianade do, anyị ga-agwa gị banyere ma e nwere contraindications ego ahụ ga-abụ na ihe omume nke ihe ovadozu, Otú ọ dị ya nwere pharmacological Njirimara, na na.
The mejupụtara nakwa ụdị ọgwụ ntọhapụ
Na ihe ụdị ike ịzụta ọgwụ "Fliksotid" ntuziaka maka ojiji nke a ga-mmasị ka owuwu? Ugbu a, ndị ọgwụ ọjọọ na-na-ere ụdị ihe inhalation aerosol. Isi nọ n'ọrụ umi bụ fluticasone propionate mikroionizirovanny. ọgwụ na-agụnye ndị dị otú ahụ ihe ọzọ akụrụngwa dị ka tetrafluoroethane.
Emepụta metal agwọ ọrịa inhaler nke nwere a concave ala na a metering ngwaọrụ onwem na a sprayer. Inside akpa bụ a nkwusioru nke na-acha ọcha ma ọ bụ fọrọ nke nta na-acha ọcha. Na Ịzụ nke ngwaọrụ, jide n'aka na ntị ka elu nke inhaler. Ya valvụ enwela anya ntụpọ.
Types of aerosolized ọgwụ
Dabere na ókè nke na-arụsi ọrụ ike mgwa ihe bụ ugbu a na nkwusioru, e nwere atọ ụdị ahụ nọchiri anya ya agwọ ọrịa. Aha ha na-agụ dị ka ndị a: "Flixotide discus", "Fliksotid Nebula" na "Flixotide Evohaler."
The pharmacological e ji mara nke ọgwụ
Gịnị bụ ọgwụ "Fliksotid"? Ntuziaka maka ojiji na-ekwu na ya nọ n'ọrụ mmewere na-ezo aka otu GCS obodo mmetụta. Mgbe ndinọ site inhalation n'ọrụ umi-arụpụta akpọ antiallergic na antiinflammatory mmetụta. N'ihi ya, dị ịrịba belata ogo mgbaàmà, nakwa dị ka ugboro nke exacerbations pathologies esonyere airway mgbochi (e.g., ala ala bronchitis, ụkwara ume ọkụ na emphysema).
The na-arụ ọrụ ụkpụrụ nke ọgwụ (aerosol)
Olee otú ọgwụ "Fliksotid Nebula" na ụdị ndị ọzọ nke a ọgwụ? Ihe bụ isi umi nke ibelata poolu cell proliferation, macrophages, eosinophils, neutrophils na lymphocytes nakwa dị ka ebelata mmepụta ma hapụ ndị ogbugbo nke mbufụt na ndị ọzọ biologically ifịk bekee (dị ka histamine, prostaglandin, leukotriene, a cytokine).
Na-adịghị ala ala okpo ọrịa akpa ume elu nrụpụta mmetụta nke a ọgwụ na-arụ ọrụ ngwa nke akụkụ okuku ume na usoro, n'ihi na ọrịa mgbaàmà-adịghị dị ka akpọ, ugboro na ogo nke exacerbations na-ebelata, na-ọ dịghị mkpa na-extra GCS mbadamba. N'ihi ya, ọ enwekwu àgwà nke ndụ nke onye ọrịa.
Systemic edinam nke ọgwụ owụt minimally. Na nke a, na ọgwụgwọ doses, ọ fọrọ nke nta ka ọ dịghị utịp ke hypothalamic-pituitary-adrenal axis.
Agwọ ọrịa "Fliksotid", nke analogues ga-aha n'okpuru ebe a, ngwa ngwa weghachiri ọrịa omume bronchodilators, na-ebelata ugboro ole nke ha were.
The ọgwụgwọ mmetụta mgbe ngwa nke aerosol inhaler amalite n'ime ụbọchị na esịmde a kacha izu abụọ ma ọ bụ karịa. N'ihi na-echekwara maka ọtụtụ ụbọchị mgbe discontinuation nke ọgwụ.
The pharmacokinetics nke aerosolized gị n'ụlọnga
Mgbe aerosol "Fliksotid" e ji mee ihe maka ya bipụta ya, nzube ya, kpam kpam bioavailability nke nọ n'ọrụ umi bụ 8-11%.
Systemic ọgwụ absorption emee isi na ngụgụ. Site n'ụzọ, ibido na absorption a rụrụ ngwa ngwa na mgbe ahụ na slows ala. N'oge usoro, akụkụ nke kuru nkwusioru nwere ike loro onye ọrịa. Otú ọ dị, ya systemic ikpughe bụ ntakiri n'ihi ndị ogbenye solubility nke ọgwụ na mmiri, dị ka nke ọma dị ka ọtụtụ metabolism dị ka ọ na-agabiga imeju.
Plasma protein nkịtị nke ọgwụ na a moderately elu na bụ banyere 91%. Active ọgwụ na-metabolized na imeju mmewere metụtara CYP3A4. N'ihi ya, na-adịghị ejekwa metabolites ii.
Agwọ ọrịa "Fliksotid" nke ukwuu n'ime nti reviews, nwere a pụtara elu plasma nwechapụ. N'oge ya ọkara ndụ bụ banyere 8 awa. Mmepụta ya dị ka metabolites na mmamịrị.
Egosi maka ojiji nke aerosol n'aka
Mgbe ụfọdụ, na-amalite "Fliksotid" ọgwụ ọjọọ? Ntuziaka na ngwa na-akọ na ndị ọgwụ kenyere maka ọgwụgwọ nke ọrịa ndị na-ata ahụhụ site na ụkwara ume ọkụ, eru dị arọ ma ọ bụ agafeghị oke ụdị. Ọzọkwa, agwọ ọrịa na-eji maka na-egbochi ọgụ mgbe anata systemic corticosteroids.
Ọzọkwa, agwọ ọrịa na-owụt ke ọrịa na-adịghị ala ala akpa ume ọrịa. Jiri ya iji belata bronchial mgbochi, nakwa dị ka mma ventilashion nke akụkụ okuku ume na akụkụ.
Contraindications ojiji nke aerosol n'aka
N'okpuru ọ bụla ọnọdụ ọ bụla ikpe nwere ike ọ gaghị eji inhaler 'Flixotide'? Contraindications ndị na-esonụ ihe:
- ndidi hypersensitivity ọ bụla akụrụngwa nke agwọ ọrịa;
- nnukwu bronchospasm;
- asthmatic ọnọdụ (dị ka a mbụ n'aka);
- ruo 1 afọ.
Ọ kwesịkwara kwuru na nke a ọgwụ ọjọọ abụghị na-achọsi ike iji maka enyemaka nke ụkwara ume ọkụ ọgụ.
Imefusi ọgwụ
ọgwụ ọjọọ, "Fliksotid" nnọọ nlezianya họpụtara N'ọnọdụ dị aṅaa? Nyocha dọkịta na-ekwu na ngwá ọrụ kwesịrị ka a na-eji n'okpuru nditịm achịkwa ọkachamara na glaucoma, imeju imeju, akpa ume ụkwara nta, hypothyroidism, afọ ime, systemic na-efe efe (nje, fungal, parasitic ma ọ bụ malitere ịrịa) na lactation na osteoporosis.
Drug "Fliksotid" inhalation: ntụziaka
Dabere ụdị nke ngwaahịa, ya ojiji na onunu ogwu nwere ike iche iche. Ka ihe atụ, iji nweta ezi mmetụta, ịgba 'Flixotide discus "ga-eji mgbe niile, ọbụna mgbe kwụsịtụkwara.
Na oge nke ọgwụ na ezigbo dose nke ọgwụ kwesịrị naanị kọwaa dọkịta, na-ewere n'ime akaụntụ ọrịa na-arịa na mkpokọta adakarị picture. N'ihi na ndị okenye, na onunu ogwu bụ 100-1000 mg 2 ugboro n'ụbọchị. The ojiji nke ọgwụ na-amalite kacha nta mpịakọta na-amị a ọgwụgwọ mmetụta. Ọ bụrụ na ọ dị mkpa, na ego nke iwesa ọgwụ ọjọọ nwere ike mụbara. The kacha dose ekwesịghị gafere 2000 micrograms.
Agwọ ọrịa "Fliksotid" maka ụmụaka si 4 afọ na-ata ahụhụ site na bronchial ụkwara ume ọkụ, a na-kenyere na ego nke 50-100 mg ugboro abụọ n'ụbọchị. Ọ bụrụ na ọ dị mkpa, nke a onunu ogwu na-eji nwayọọ nwayọọ na ụba ruo 400 micrograms kwa ụbọchị. Dị ka n'ihi na ndị okenye na-adịghị ala ala akpa ume ọrịa, ha na-emekarị nyere 500 mg nke ọgwụ ugboro abụọ n'ụbọchị.
Olee otú iji ndị ọgwụ ọjọọ, "Flixotide Evohaler"?
Ngwá ọrụ a ga-eji mgbe nile. ọ na-atụ aro ịgba ọtụtụ ugboro tupu n'itinye ọgwụ maka a edo dose. Ọzọkwa, slurry dị mkpa ịma jijiji na karama. Mgbe spraying aerosol onye ọrịa a chọrọ iji mee ka a ngwa ngwa ume. Ekwuchite kwesịrị kpochara dịkarịa ala otu izu.
Olee otú iji na-atụ aro ego nke ọgwụ "Fliksotid"? Doses nke ọgwụ gbakọọ dị ka ndị a: otu-apụ ego nke ọgwụ kwekọrọ ekwekọ na abụọ sputtering.
Na bronchial ụkwara ume ọkụ na ndị okenye inye 100-1000 micrograms nke nọ n'ọrụ umi ugboro abụọ n'ụbọchị. The ojiji nke ọgwụ ga-malitere na ala irè doses, vposlestvii, ma ọ bụrụ na ọ dị mkpa edemede, ha nwere ike mụbara. Karịa ego nke ọgwụ ga-2000 micrograms.
Olee otú na-emeso ụmụaka iji ịgba "Fliksotid"? Inhalation ụmụ karịrị afọ anọ na ọrịa a dị ka ụkwara ume ọkụ, na-ekenye na ego nke 50-100 mg ugboro abụọ n'ụbọchị. Ọ bụrụ na ọ dị mkpa, ndị dose nwere ike jiri nwayọọ nwayọọ na ụba. Karịa ego nke oriri nke ọgwụ maka ụmụ afọ anọ bụ 400 mg.
Ndị okenye na-adịghị ala ala okpo ọrịa akpa ume ọgwụ inye 500 micrograms ugboro abụọ kwa ụbọchị. Ọ bụrụ na mgbe 3-6 ọnwa mgbe nnabata nke ọgwụ ka mma na ọ bụghị hụrụ, ọ dị mkpa ịgbanwe ọgwụgwọ Usoro.
Ọ bụrụ na a na nwa n'agbata afọ 1 na 4 afọ chọpụtara na ụkwara ume ọkụ, ọ na-kenyere 100 mg nke ọgwụ ugboro abụọ n'ụbọchị. Na nke a, inhalation na-atụ aro iji ụmụaka Spicer na-akpali aha "Bebihaler".
Aerosol "Fliksotid Nebula": ntuziaka maka ojiji
Nke a agwọ ọrịa ga-eji na-edeghị ede (na ọnụ na-ekwuru) ma ọ bụ ọ dịghị òkè (n'ihu nkpuchi) inhalation. Ọzọkwa, ọgwụ na-họpụtara dị ka ndị aerosol ugboelu nebulizer. Ọ bụ oké na-achọsi ike iji ultrasonic ngwaọrụ.
Ọ bụrụ na chọrọ ẹkama ochichi nke mmadụ ma ọ bụ ochichi nke nta doses nke agwọ ọrịa tupu inhalation usoro na-atụ aro na itughari ngwọta nke sodium chloride.
Okenye na-eto eto n'elu 16 afọ nke ọgwụ ndinọ ke ichekwa 0.5-2 mg ugboro abụọ kwa ụbọchị. The kacha onunu ogwu ga-agbasoriri maka a izu mgbe agha nke ụkwara ume ọkụ, na mgbe ahụ na-eji nwayọọ nwayọọ belata ya.
Ọ bụrụ na mmetụta nke rụọ ọrụ ndị ọnọdụ ka mgbanwe site ọgwụ "Fliksotid Nebula", nke ntụziaka mgbe nile ka ndị ọzọ na ụdị ọgwụ.
Child si 4 16 afọ agwọ ọrịa ndinọ ke ichekwa 1 mg ugboro abụọ n'ụbọchị.
ikpe nke ovadozu
Bụrụ na nke ovadozu, onye ọrịa nwere ike a nwa oge suppression nke ọrụ nke hypothalamic-pituitary-adrenal usoro, ịrịba suppression nke adrenocortical ọrụ, nnukwu adrenal nsogbu ụmụaka ndị natara a dose nke 1000 mcg kwa ụbọchị na n'elu.
Ke adianade do, ọrịa nwere dara mbà n'obi nsụhọ, e nwere apịajighị apịaji na hypoglycaemia. Ọ kwesịkwara kwuru na nnukwu adrenal nsogbu na-emekarị na-amalite na ndabere nke ọnọdụ ndị dị otú ahụ dị ka oké trauma, ịwa, ọrịa na ọnụnọ nke a nkọ ọnụ ke ọgwụ onunu ogwu.
mmetụta
Nwere ike a na-adịghị mma mmetụta na ahụ ike nke onye ọrịa n'ikuku "Fliksotid" ọgwụ ọjọọ? Mmetụta ndị fọrọ nke nta niile ngwaọrụ ahụike. Na ngosi nke kuru na nkà mmụta ọgwụ na-adịghị ma e wezụga.
- Dịghịzi usoro: akpụkpọ Jeremaya mere n'ihi hypersensitivity, angioedema (oropharynx na ihu), ọrịa nke akụkụ okuku ume usoro (dyspnea ma ọ bụ bronchospasm), anaphylactic ujo.
- Na parasitic na-efe efe: candidiasis ọnụ na akpịrị, na thrush. Dị otú ahụ na abnormalities na-atụ aro ka itucha akpịrị na ọnụ na mmiri nkịtị. Ọ nwekwara ike-eji antifungals obodo edinam. Nnọọ nkịtị mmetụta na-esonụ na ojiji nke aerosol bụ oyi baa, ma naanị na ọrịa na COPD.
- Metabolism: hyperglycemia.
- Endocrine usoro: Cushing si syndrome, ịda mbà n'obi ime ihe nke adrenal cortex, belata mineralization nke ọkpụkpụ anụ ahụ, ibu iberibe, cataracts, glaucoma.
- Ụjọ usoro: nchegbu, akparamàgwà ọrịa, na-ehi ụra, ahụ mgbakasị na hyperactivity (karịsịa ụmụ).
- Subcutaneous abụba: ichihịa.
- Akụkụ okuku ume na usoro: hoarseness (na-atụ aro ozugbo usoro na ikwacha akpiri gị ọnụ mmiri), paradoxical bronchospasm.
Adọ aka ná ntị mgbe eji ọgwụ
Inikiet inikiet kagbuo na ojiji nke ọgwụ ọjọọ na-adịghị atụ aro.
Karịsịa ịkpachara anya na ọgwụgwọ nke kuru corticosteroids na ọrịa na-adịghị ejekwa ozi ma ọ bụ ike n'ụdị ụkwara nta.
Ịgbaso oru nke ọgwụ ndị dọkịta ga-elele na onye ọrịa maara otú iji ihe inhaler. N'oge usoro, ọ dị mkpa iji hụ na Mbelata nke ọgwụ na ihe na-ewe ebe mmekọrịta na ume. Naanị otú a na-enwe ndidi ga-enwe ike iji hụ na ezigbo nnyefe nke nọ n'ọrụ mmewere ngụgụ.
Ọ na-atụ aro ka nọgidere nyochaa Ọnọdụ nke uto nke-eto eto ụmụ na-anata kuru corticosteroids maka a ogologo oge.
Mgbe na-ebufe ọrịa site na ịnweta systemic corticosteroids maka inhalation ọgwụ nwere ike njọ anabata ọrịa na (e.g., imi nsụchi ma ọ bụ eczema) na mbụ-ewute systemic ọgwụ. N'ọnọdụ dị otú ahụ, symptomatic ọgwụ na Antihistamines ma ọ bụ Nde ọgwụ.
Dị ka ọtụtụ kuru ọgwụ na aerosol containers, na ọgwụgwọ mmetụta nwere ike belata mgbe obi jụrụ ịgba.
Iji ụbọchị, e nwere obere akụkọ na-enwe ndidi, anyị na-atụle na-eji ngwá ọrụ, na-abawanye na ọbara glucose etoju. Nke a mgbe niile kwesịrị icheta dọkịta mgbe prescribing ọgwụ ka ọrịa na-arịa ọrịa shuga.
Mmetụta nke nọ n'ọrụ umi ke a onye nwere ikike iji rụọ ọrụ na igwe na-arụ ọrụ na ígwè ọrụ ndị na-achọ elu ịta, eleghi anya.
Analogs agwọ ọrịa
Gịnị ọgwụ zuo, ma ọ bụrụ na onye ọrịa ahụ na-enwe ike ịzụta ọgwụ "Fliksotid"? Analogs nke ngwá ọrụ nwere n'ụzọ otu Njirimara. Ma tupu n'itinye ha nwere ike ikwu na ị na-agụ nchọ ntụziaka, nakwa ịkpọ a ọkachamara.
Ugbu a, ndị na-esonụ analogue nke ọgwụ: ọgwụ ọjọọ "Kutiveyt", "Nazarel" "Flixonase" "Fluticasone" na "Valium." Ọ ga-kwuru na price nke ndị a ọgwụ ọjọọ nwere ike ịbụ dị iche iche karịa mbụ. Site n'ụzọ, na aerosol "Fliksotid" i nwere ike ịzụta n'ihi na 570 (50 .mu.g, 120 doses), 840 (125 mg, 60 doses) ma ọ bụ 140 (250 .mu.g, 60 doses) Russian rubles.
Nyocha nke-eji imi ekuru
Gịnị na-eme ndị dọkịta na ndị ọrịa banyere ọgwụ 'Flixotide'? Nyocha nke a owuwu ndị tumadi mma. Nke a bụ n'ihi bụ isi eziokwu ahụ bụ na aerosolized agwọ ọrịa nwere dịtụ elu arụmọrụ. Ọ budata ebelata ugboro nke ọgụ nke ọrịa na ụkwara ume ọkụ, na mma bronchial patency na ndị na-ata ahụhụ si na-adịghị ala ala akpa ume ọrịa.
Ma ihe ndị na-ezighị ezi reviews, dị ka a na-achị, ha na-abịa site na ọrịa ndị na-eji ọgwụ ọhụma ma ọ bụ adịghị kenyere a dọkịta. Ya mere, iji nweta ihe ndị kasị mma na-arụpụta n'ihu iji ọgwụ, nakwa dị ka ya ogbo, ọ na-atụ aro ka na-amụ na zuru ezu na nchọ ntuziaka maka ojiji. Ọzọkwa, ọ dị oké mkpa ka ha hụ dọkịta, onye na, n'eziokwu, na ga nwere ike ikwu na ngwá ọrụ a, dabere na ihe ike na ule.
Olee otú iji chekwaa aerosol Nwa?
Kuru aerosol na-atụ aro ka na a gbara ọchịchịrị ebe okpomọkụ adịghị gafere 25 degrees. Adị ndụ nke ọgwụ bụ kpọmkwem afọ abụọ. Mgbe oge a ọ na-aju iji.
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