Ahụ ike, Preparations
Ntuziaka maka ojiji "tiapridal". Analogs na reviews
"Tiapridal" - antipsychotic ọgwụ arụpụtara site tiapride. The ọgwụ na-etinyere ka a ogwuura, analgesic na hypnotic. Ndabere nke antipsychotic edinam - igbochi dopamine anabata, nke budata emetụta ịrụ ọrụ nke CNS. N'isiokwu a anyị na-akọwa n'ụzọ zuru ezu banyere ọgwụ.
Mejupụtara gụnyere ọgwụ
The na nkà mmụta ọgwụ dị na abụọ iche-iche, na mbadamba nwere ike zụrụ na ngwọta:
- Otu mbadamba dị ka otu ampoule mejupụtara 100 milligrams nke isi akụrụngwa na inyeaka bekee. Inyeaka Efrata eji na mejupụtara nke povidone, magnesium stearate, mannitol. The mejupụtara na-gbakwunyere na otu okenye colloidal dioxide, sịlịkọn na microcrystalline cellulose.
- E wezụga isi akụrụngwa nke ngwọta mejupụtara sodium chloride na mmiri ogwu ogbugba.
Na otu igbe nwere 20 mbadamba (2 blisters na 10 mbadamba) ma ọ bụ 12 vials (2 blisters nke 6 vials). Ntuziaka maka ojiji "Tiapridal" n'ụdị nke a ngwọta maka ọgwụ na-enye ohere ndinọ intravenously na intramuscularly. Nke a na ụdị ọgwụ bụ naanị ndị kwesịrị ekwesị maka ọgwụgwọ nke okenye ọrịa.
Pharmacodynamics "tiapridal"
The agwọ ọrịa nwere neuroleptic, analgesic na anxiolytic edinam. Dị ka ntụziaka ntuziaka, "Tiapridal" bibiri nkanka ịrụ ọrụ nke D 2 anabata nke Central dopamine. N'ihi ya na D 1 anabata nwere dịghị mmetụta. The ọgwụ ego n'anya Bibie nke psoriasis, mgbe eji na ndị agadi mma na-eche echiche.
Pharmacokinetics "tiapridal"
Intramuscular ochichi nke ọgwụ (200 mg) nke ya kacha larịị ke idem achọpụtara mgbe 30 nkeji, na-eji mbadamba n'otu dose - 60 nkeji. The bioavailability nke ọgwụ mgbe eji ozugbo tupu nri na 75% ụba 95%. N'ihi na ọgwụ ọjọọ ndị dị otú ahụ were na-abawanye na ya kacha larịị na organism (40%).
Absorption ke idem bụ iji nwayọọ na agadi ọrịa. "Tiapridal" ntuziaka maka ojiji na-ezo aka ihe gị n'ụlọnga obe na placental na ọbara-ụbụrụ mgbochi. Ọ maara na n'oge na ọgwụgwọ na ọgwụ bụ ugbu a na ihe ndị mejupụtara nke mmiri ara. Na ndị inyom, ele mmadụ anya n'ihu mwepụ nke ọgwụ ngwa ngwa karịa na nke ndị ikom (ihe karịrị 2.9 awa), ihe dị iche bụ 0,7 awa. Metabolism ji dị ka agafeghị oke. Isi akụkụ nke ọgwụ (70%) na-ewepụ ahu site na akụrụ na-agbanweghi agbanwe.
Egosi "Tiapridal" nkwadebe
Mejuputa ọgwụ na ọgwụ ọjọọ "Tiapridal" ọgụgụ dị ka ndị a:
- dyskinesia (tardive, n'amaghi ama);
- Gilles de la Tourette syndrome;
- chorea;
- akparamàgwà ọrịa (ike ike na steeti, n'ahụhụ et al.), dapụtara na a ọkpụrụkpụ eruba nke-adịghị ala ala aṅụrụma na ndị agadi ndị ọrịa;
- na-adịghị mma ngosipụta na omume, dị ka ike ike ikwu na n'ahụhụ;
- mgbu kpụ ọkụ n'ọnụ agwa (-adịghị ala ala ụdị).
Contraindications, na-agaghị emeli na-enweta "Tiapridal" ọgwụ
Machibidoro imposition nke "Tiapridal" ntuziaka maka ojiji maka ụmụ onye afọ bụ ihe na-erughị afọ isii. Na ụmụaka ọgwụ a rụrụ naanị mkpụrụ ọgwụ. The ọgwụ na-ekwesịghị-emeso ụmụ nwaanyị dị ime na ndị ọrịa bụ ndị na-ara. Ọgwụ na-adịghị mee bụrụ na nke hypersensitivity ka ya mmiri, na ndị ọzọ dị otú ahụ. Contraindications gụnyere ekwu, sị:
- hepatic na gbasara akụrụ odida, nke nwere bukwanu ogo;
- prolaktinzavisimogo Ịchọpụta Otú Nsogbu etuto ahụ, enyo nke ya edidu;
- hypertensive nsogbu;
- nchoputa nke pheochromocytoma, a enyo nke ya adị.
Mbadamba na ihe ngwọta na-eji na "sultopride" na dopamine ihe nnabata agonists (e wezụga bụ ọgwụgwọ nke ọrịa na ọrịa Parkinson) na-adịghị jikọtara na ụdị ụfọdụ nke neuroleptics, mgbochi arrhythmic mmadụ nke klas m na III A.
Medicating "Tiapridal" ntụziaka adịghị ekwe ka n'out oge na-eji "Moxifloxacin", "sparfloxacin", "Difemanila", "Erythromycin", "bepridil," "mizolastine", "levodopa", "cisapride" na na igba ogwu n'akwara "vincamine" .
Ọ bụrụ na onye ọrịa (karịsịa ndị agadi) na-emeso-eji ọgwụ ọjọọ nwere ike na-eduga mmepe nke hypokalemia, gbasara obi conduction arịa ọrịa, amụba QT nkeji, omume nke bradycardia owụt agwa, na-eji "Tiapridal" ga-ọma. Ịkpachara anya a chọrọ dị otú ahụ ikpe:
- Ọrịa Parkinson;
- congenital QT nkeji elongation agwa;
- hypokalemia;
- adịghị ala ala gbasara akụrụ odida;
- bradycardia;
- ọrịa na nke akwusila obi usoro (decompensation nzọụkwụ);
- Akwụkwụ na-adọ.
Ọgwụgwọ na "Tiapridal"
na ngwa nke "Tiapridal" ntuziaka tụrụ aro iji a mbụ na obere doses, nke nta nke nta na-amụba ha, iji nweta karịa mmetụta.
akparamàgwà ọrịa
N'ihi na ha onwe dị mkpa itinye 200 mg nke ọgwụ kwa ụbọchị (ruo 300). The mmetụta dị mma a na-enweta na izu isii na nkezi. Older ọrịa ndinọ a ala dose ọgwụ - 50 mg. A otu dose kwesịrị gwusia ugboro abụọ n'ụbọchị, na ya na-abawanye na-kwere na ngakọrịta nke kwuru kpọmkwem nkeji, ihe ahụ a rụrụ nwayọọ nwayọọ, na-echebara ọkachamara ndụmọdụ. The kwa ụbọchị dose ekwesịghị gafere 300 mg.
-Adịghị ala ala na-ufiop mgbu
The kwa ụbọchị dose nke ọgwụ maka ọgwụgwọ nke ọnọdụ ndị dị otú bụ site na 200 na 400 mg.
Chorea, Gilles de la Tourette syndrome
Mgbe arụ ọgwụgwọ nke nwa kwa ụbọchị dose họrọ-ewere n'ime akaụntụ arọ ahụ na banyere 3-6 mg / n'arọ. Ọ bụrụ na ị mkpa ka o duzie ihe okenye ọrịa, mbụ ji mee 25 mg nke ọgwụ kwa ụbọchị, mgbe e mesịrị (mgbe a nwayọọ nwayọọ na-abawanye na dose) - 300-800 mg.
Oyobio, ime ike ike
The aro ya kwa ụbọchị dose nke agwọ ọrịa bụ site na 100 na 150 mg.
akparamàgwà ọrịa
The na-atụ aro dose maka n'ehihie ojiji (site na 200 na 300 mg) na ihe banyere delirious ekwu ma ọ bụ predelirioznogo adahade 400-1200 mg. The kacha ekwe omume dose nke gaghị karịa, bụ 1800 mg. The mmeghe nke ọgwụ na-emepụta na nkezi ise ọ bụla awa. Ọ bụrụ na ọgwụgwọ dị mkpa ka ndị agadi onye, ụbọchị ọ bụla bụ 2-3 injections n'agbata nke hụrụ nkeji nke 6 awa. Maka ọgwụgwọ nke ndị dị otú ahụ ọrịa na-atụ aro ya kwa ụbọchị oriri nke 200 na 300 mg nke agwọ ọrịa na a oge na-ekwe ka tinye ihe na-erughị 100 mg "tiapridal".
Ufiop ngosipụta nke a na-adịghị ala ọdịdị nke ihe mgbu
Ọgwụgwọ dabeere na ndinọ kwa ụbọchị dose kwekọrọ 200-400 mg nke ọgwụ.
Mmetụta mgbe na-ewere "Tiapridal" ọgwụ
Mgbe n'imeso ọgwụ "Tiapridal" ntụziaka ntuziaka, reviews n'ịkwado likelihood nke ụfọdụ oghom Jeremaya mere. Mebiri nwere ike ime na urogenital, ụjọ, endocrine na obi usoro. Ọzọkwa, e nwere ihe ize ndụ nke nsogbu na uche ziri ezi. N'ihi na ndị ọzọ mmetụta ọjọọ na-agụnye allergies, anụ ngosipụta esonyere ibu ibu, orthostatic hypotension.
Ovadozu "tiapridal"
Ọ bụrụ na ị na-eji oké dose omume ovadozu na ya bụ ọrịa bụ na-enwe nsogbu nke nsụhọ, ndị kasị njọ nke na - Coma, neuroleptic syndrome (ịza aza, nnukwu forms). Iji dozie a ala nke organism a rụrụ ọgwụgwọ dabeere anticholinergic mmadụ. Mgbe abolition nke ọgwụ dị mkpa na-ebu symptomatic ọgwụgwọ na plasmapheresis.
adọ aka ná ntị
Tupu were a na nkà mmụta ọgwụ "Tiapridal" ntụziaka ntuziaka na-atụ aro na ị na-agbazi hypokalemia. N'oge ọgwụ ọ dị mkpa ka mgbe niile nyochaa electrolyte itule, na-eduzi ihe ngwá, nyochaa adakarị picture mgbanwe.
Ọ bụrụ na ọ dị mkpa itinye anticholinergic ọgwụ ọjọọ eme anata neuroleptics extrapyramidal syndrome mepụtara kama dopamine ihe nnabata agonist.
Mgbe oge nke ọgwụgwọ hapụ omume ndị na-abụrụ a pụrụ iyi egwu, ọ na-adịghị na-atụ aro na-arụ ọrụ nke chọrọ pụrụ iche na-elekọta ma ngwa ngwa.
Mmekọrịta ndị ọzọ bekee
Ụfọdụ Nchikota preparations na-ewere ọgwụ "Tiapridal" ntụziaka, nzaghachi metụtara na puru nke omume nke undesired Jeremaya mere. Ọ na-adịghị na-atụ aro mgbe ọgwụgwọ etinyere "Clonidine", Antihistamines, anxiolytics, barbiturates na opioids, dị ka "tiapridal" mmetụta ga-akpọ. N'ihi incompatibility ghara iwere "levodopa" na-aba n'anya. Ọgwụ nwere ike ikpokọta na ojiji nke neurotrophic ọgwụ ọjọọ, analgesics, antidepressants, neuroleptics. Elu n'ihe ize ndụ nke orthostatic hypotension, e nwere n'otu oge ojiji nke antihypertensive ọgwụ ọjọọ na "Tiapridalom".
The na-eri nke ọgwụ ọjọọ na analogues, reviews banyere ọgwụ ọjọọ, "Tiapridal"
Ọ bụrụ na ọ dị mkpa ọgwụgwọ "Tiapridal" pụtara ntụziaka nkọwa ka ị mara ihe a ọgwụ bụ. The price nke ọgwụ ọjọọ dị mkpa nke ukwuu na nhọrọ nke a agwọ ọrịa n'ihi na ọgwụgwọ. The ngwọta na vials nwere ike zụta maka banyere 995 rubles, na mbadamba - maka 1,400 rubles.
N'etiti analogues nke ọgwụ - "Eglonil", "Betamax". Nke ndị nọ n'ọnọdụ nwere ike họrọ "Sulpiride" ma ọ bụ "Prosulpin". E nwere ihe ọzọ analogue nke ọgwụ - "tiaprid", ọ na-atụle ihe ndị kasị mfe inweta, ọ bụ nnọọ ihe a na-ewu ewu nhọrọ, na anụ ụlọ ọgwụ mmepụta nke na-emekọ na ụlọ ọrụ "Organic". Dị ka akụkụ nke "tiaprid" chee otu ifịk umi, nke bụ akụkụ nke ọgwụ "Tiapridal". Ojiji analogs Guide na-atụ aro iji họrọ, mgbe mbụ apụghị-eji n'out oge na ụfọdụ ọgwụ ọjọọ na-eme ka mmetụta na-adịghị na-enye a chọrọ mmetụta. Iji ọgwụ kasị irè, gaa na akaụntụ ọtụtụ n'ime ihe mgbe họrọ.
N'oge ọgwụgwọ, ọ dị mkpa na-eso niile ihe dọkịta gwara na-atụ aro, bụ nke nwere ntuziaka maka ojiji. "Tiapridal", dị ka e gosiri site nzaghachi, ọtụtụ mgbe, a na-eji wepụ ọnọdụ so site ụjọ ụtọ, na-eme ihe ike ike omume, mmanya psychosis. Na-emekarị, ndị ọrịa na dọkịta nwere afọ ojuju na n'ihi nke ọgwụ. Ihu ọma, a ala mmuta bụ chọrọ n'ihi na ezi mmetụta na-emepe emepe mgbe mmejuputa mbụ N'ezie. Nyocha na-egosi na ọrịa na nkà mmụta ọgwụ "Tiapridal" mfe iji.
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