Ahụ ike, Preparations
Ọgwụ "Buspirone": reviews nke dọkịta
ma ọgwụ dị irè "Buspirone"? Ọbịa, bụ ndị kpọọrọ ngwá ọrụ a ga-ọkọnọ n'okpuru. Anyị na-agwa gị banyere ihe Njirimara nke si ọgwụ ikpe nke ọ họpụtara, ma ọ bụrụ na o nwere ọ bụla contraindications na mmetụta.
Na udi ma na mejupụtara nke ọgwụ
Ihe e lere a "buspirone" ọgwụ ọjọọ? Nyocha nke dọkịta na-ekwu otú ahụ arụ ọrụ bekee ndị dị otú ahụ dị ka buspirone hydrochloride. Ke adianade do, agwọ ọrịa nwere ihe ọzọ mmiri n'ụdị lactose, ọka starch, calcium hydrogen phosphate dihydrate, starch (ụdị A), sodium, colloidal sịlịkọn dioxide, magnesium stearate na MCC.
Dị bụ ngwá ọrụ na ụdị-acha ọcha, gburugburu mbadamba enịm ke a ikpo nke kaadiboodu.
The pharmacodynamic Njirimara nke ọgwụ
Gịnị Njirimara nke ọgwụ "Buspirone"? Ntuziaka, comments dọkịta agwa ọrịa banyere ihe bụ ihe anxiolytic ọgwụ. Ọ na-zubere maka ọgwụgwọ nke nchegbu ọrịa dị iche iche si malite.
The kpọmkwem usoro nke ihe nke mbadamba na-adịghị arụnyere. Otú ọ dị, ndị ọkachamara na-arụ ụka na ọgwụ bụ a nhọrọ agonist na postsynaptic 5-HT 1a anabata na ụjọ usoro.
Mgbe na-ewere ọgwụ ọjọọ na-eji nwayọọ nwayọọ na-egosipụta ya edinam. Mmetụta nwere ike hụrụ n'ihi na otu onye ka izu abụọ. The kacha ọgwụgwọ mmetụta chọpụtara na mgbe a ọnwa.
The pharmacokinetic Njirimara nke ọgwụ
Ebe absorption nke ọgwụ "Buspirone"? Ọbịa ọkachamara na-atụ aro na a ọgwụ nnọọ ngwa ngwa na fọrọ nke nta kpamkpam etinye obi gị dum na eriri afọ tract. The plasma ọgwụ ịta hụrụ mgbe 1-1.5 awa. Communication na-edozi bụ 95% na nkera ndụ - awa atọ.
Odika 30-65% nke nọ n'ọrụ mgwa na ya metabolites na-anyụpụ na mmamịrị n'oge ụbọchị na 20-40% na-egosipụta ọnụ na na nsị. Ọ bụrụ na onye ọrịa nwere nsogbu na imeju na-na akụrụ ha mkpochapu mbelata ubé.
Egosi maka ojiji nke mbadamba
Maka nzube dị otú ahụ a ọgwụ dị ka "Buspirone" nwere ike a ga-amanye? Nyocha nke dọkịta na-ekwu na a ọgwụ na-eji na ọnụnọ nke nchegbu ọrịa na-ebu mgbaàmà ndị dị otú ahụ dị ka nchegbu, nchegbu, na ubara nchegbu.
Contraindications ojiji nke ọgwụ
Gịnị na-ọnọdụ nke onye ọrịa a machibidoro iwu na-ọgwụ "Buspirone"? Ọbịa ọkachamara na-ekwu na ọgwụ na-ekwesịghị kenyere ndị na hypersensitivity ka ndị bụ isi na ndị ọzọ bekee ọgwụ ọjọọ, myasthenia gravis, nnukwu congestive glaucoma, oké gbasara akụrụ impairment, Akwụkwụ na-adọ na oké imeju dysfunction.
Ọzọkwa, tụlee ọgwụ na-contraindicated na ụmụaka na n'oge ara.
Drug "Buspirone": ntuziaka maka ojiji
Comments banyere nke a na nkà mmụta ọgwụ ga-ọkọnọ a obere n'ihu.
The Regulations weghaara na agwọ ọrịa, na-akọ na dose ga-họọrọ naanị site na ịga dibịa, dabere na ọrịa na-arịa.
Na-emekarị, na mmalite nke ọgwụ ọgwụgwọ a na ndinọ ego nke ise milligrams ugboro atọ n'ụbọchị. Kwuru nwayọọ nwayọọ dịkwuo dose ka 15-30 mg (partitioned n'ime ọtụtụ doses).
The kacha kwa onunu ogwu nke ọgwụ ekwesịghị ịbụ ihe karịrị 45 mg, na otu - adịghị karịa 30 mg.
Olee otú m ga-ewe "Buspirone"? Ntụziaka na-ekwu na-edu mkpụrụ ọgwụ kwesịrị ụbọchị ọ bụla n'otu oge. Ha apụghị ata. The ọgwụ kwesịrị naanị aṅụ a obere ego mmiri.
Ndị na-mkpọchị ọrụ nke akụrụ ma ọ bụ imeju kwesịrị na-kasị ala-ekwe omume usoro onunu ogwu.
Duration nke N'ezie kpebisiri ike n'otu n'otu (ikpe site ikpe). A machibidoro iwu na-ọgwụ ruo ogologo oge, karịsịa enweghị nlekọta nke ndị ọrụ.
Ke ukem na ọgwụgwọ na-atụ aro sotsioterapevticheskie na psychotherapeutic jikoro.
ikpe nke ovadozu
Gịnị na-ịrịba ama nke ovadozu-eme mgbe na-ewere elu doses nke ọgwụ "Buspirone"? Ọbịa ọkachamara na-atụ aro ndị na-esonụ iche: cramps, agbọ onunu, ike ọgwụgwụ, ajụ obubu, disturbances nke afo, vomiting.
Na ovadozu gastric lavage a rụrụ, nakwa dị ka nlekota nke ọbara mgbali, respiration, na obi otiti. Ọgwụgwọ - symptomatic.
mmetụta
Ò mmetụta nke ọgwụ "Buspirone Sandoz?" Nyocha nke ọrịa na dọkịta na-atụ aro na ọgwụ pụrụ iduga nnọọ a ọnụ ọgụgụ buru ibu nke oghom ihe:
- myocardial infarction, nwa oge ọnwụ nke nsụhọ, obi ọdịda, na-abụghị kpọmkwem obi mgbu, ọrịa strok, tachycardia, bradycardia, hypotension ma ọ bụ ọbara mgbali elu, cardiomyopathy;
- conjunctivitis, bịara ikiri ọhụụ, ụjọ nke mgbali n'anya, nācha ọbara-ọbara nke na-edozi, na-egbu mgbu sensashion n'anya na ibelata ubi nke na-ele, itching, photophobia;
- ogwe, nchegbu, mkpọchị nchikota, na-arọ nrọ, extrapyramidal ọrịa, ehighi ura, n'amaghi mmegharị, ịma jijiji, mara jijiji, obi ụtọ, nsogbu nke ụda, ibu iro, mkpọchị ebe nchekwa, ịda mbà n'obi, slurred okwu, iro ụra, serotonin syndrome, dizziness, nkụnwụ, mgbada anya, stupor, mgbagwoju anya, na ọnọdụ swings, depersonalisation, claustrophobia, ụda uche, fever, hyperkinesia, mkpọchị associative nghọta, enweghị mmasị, anuri, gallyutsi mba, igbu onwe ideation, paresthesia, ọdụdọ, ọrịa Parkinson, ahụ erughị ala, lethargy, psychosis, akathisia;
- Ugboro urination, urinary njigide, abalị urination, enuresis;
- epistaxis, gọzie gị mkpọchi, mkpụmkpụ nke ume, akpịrị akpịrị, mkpụmkpụ nke ume, mkpi nke obi;
- arthralgia, isi na muscle spasm, myasthenia, myalgia;
- mgbanwe ọbara kwa;
- oyi hypersensitivity, ike ọgwụgwụ, ọchịchọ gabigara ókè oriri nke na-aba n'anya, isi ọwụwa, mkpọchị ọbara clotting, abawanye ma ọ bụ ọnụ ke arọ, na-ekpo ọkụ mgbukepụ, mmetụta nke ịkụ na isi, ihe ọkụ ọkụ, malaise, ike ọgwụgwụ, mkpọchị uto na isi, ọnwụ nke olu, hiccups, glossalgia;
- tinnitus;
- ịhụ nsọ ọrịa, na-ebelata ma ọ bụ na ụba libido, mbufụt nke urogenital akụkụ, amenorrhea, enweghi ike, belata ejaculation;
- otutu, edema, ecchymosis, hyperemia, pemphigus, alopecia, akọrọ, eczema, nfụkasị Jeremaya, urticaria, thinning nke ntu, hematoma;
- afọ ọsịsa, agbakasị bowel syndrome, salivation, ọgbụgbọ, orùrù-ọbara site na ikensi, epigastric mgbu, elu imeju enzymes, akọrọ ọnụ, afọ ntachi, flatulence, mụbara ma ọ bụ na-ebelata mmetụta nke agụụ, vomiting;
- galactorrhea, mkpọchị thyroid ọrụ, gynecomastia.
ọgwụ interactions
Tupu eji "Buspirone" ọgwụ kwesịrị ijide n'aka na-agụ ntụziaka. Ọ na-enye ndị na-esonụ ozi banyere ọgwụ interactions kwuru ọgwụ:
- Mgbe jikọtara ihe antidepressant, antihypertensive mmadụ, gbasara obi glycosides, anticoagulants, hypoglycemic na neuroleptic mmadụ nakwa dị ka ọnụ na gbochie afọ na-achọ siri ike na-achịkwa. Mmekọrịta sedatives na benzodiazepines adịghị anakwere.
- Strong inhibitors nke cytochrome P450 abawanye bioavailability "buspirone".
- Ọ na-adịghị na-atụ aro na-ọgwụ na Mao inhibitors n'ihi ihe ndị pụrụ omume nke hypertensive nsogbu.
- Ọnụ na mbanye "Cimetidine" kacha ịta "buspirone Sandoz" na-amụba site 40%.
- "Rifampicin" ebelata kacha ọgwụ ịta nke banyere 89,6%.
- Mgbe jikọtara ọgwụ ọjọọ na-emetụta nke kacha ịta nke "buspirone", ọ na-achọsi ike ka ịhazie dose nke ikpeazụ.
- "Ritonavir" na "ketoconazole" ngọngọ ndu mgbanwe "buspirone" nakwa dị ka ntọt ya plasma ịta.
- Na Nchikota ọgwụ na a "diazepam" ọdịnaya nke ikpeazụ nwere ike mụbara n'ime ọbara plasma. Ke adianade do, e nwere ike ịbụ mmetụta dị otú ahụ dị ka ọgbụgbọ, dizziness na isi ọwụwa.
- Imekotaotuugbo n'ikuku "buspirone" na "Haloperidol" pụrụ ịmụba ọbara etoju.
- Ọ kwesịrị izere aṅụ mmanya n'oge ọgwụgwọ "buspirone Sandoz."
Drug "Buspirone": testimonials nke ndị mmadụ (na-eji ọkụ) na ndị ọkachamara
Kasị ọrịa na-ahapụ mma nzaghachi banyere a ọgwụ. Ha mara na ya elu arụmọrụ. About mmetụta kọrọ nnọọ adịkarịghị.
Ọkachamara na-ekwu na-ewere mkpụrụ ọgwụ ndị a bụ nnọọ ihe na-akpatakarị ekwesighi mmetụta. Ha nwere ike na-hụrụ na a iche iche udi nke ọrịa. Na nke a, mmetụta dị naanị nwayọọ na ngwa ngwa rue enweghị discontinuation nke ọgwụ.
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