Ahụike, Nkwadebe
Tioktatsid®: analogues. Tioctacid®: ntụziaka, ọnụahịa, nyocha
Tioktatsid® bụ nkwadebe nke thioctic (nke a na-akpọkwa alpha-lipoic) acid. Alpha-lipoic acid bụ antioxidant siri ike, onye dị mkpa na ọtụtụ mmepụta ihe ndị dị ndụ na usoro nhazi ahụ na ahụ mmadụ, ebe ọ na-emepụta ya. Ọrụ nke thioctic acid bụ ichebe mkpụrụ ndụ nke ahụ site na mbibi na-emerụ ahụ nke mgbatị dị ala. Tụkwasị na nke ahụ, a na-emepụta thioctic acid ma na-ekere òkè n'ime mweghachi nke usoro antioxidant na-ahụ anya n'ime ahụ. Karịsịa, mkpụrụ alpha-lipoic acid na-akwalite mweghachi nke vitamin C na E, coenzyme Q10, mmụba nke nrịta nke njiri mmiri nke antioxidant.
Tioctacid® nwere mmetụta nootropic, na-egbochi imeju, na-ebelata ịta nke lipids n'ime ọbara, gụnyere cholesterol, na-akwalite usoro nke iji glucose eme ihe site na ahụ nke ahụ, si otú ahụ belata ọkwa ya n'ime ọbara. Ihe si na mmetụta dị otú ahụ dị mgbagwoju anya bụ mmụba nke ngosipụta nke insulin resistance nke organism. Ọzọkwa, Tioctacid® na-ebelata agụụ, na-akwalite usoro mmanu oxydation, wee si otú ahụ na-egbochi nchịkọta nke nchịkwa abụba ma na-enye aka na-emeziwanye ahụ ike, gụnyere ịgwọ oke ibu.
Tioctacid® BV (nkwụsị ngwa ngwa) bụ ọgwụ na ụdị ụdị ọgwụgwọ, kachasị mma iji were ọnụ. Ụdị a na-achọpụta na ihe ụfọdụ nke ọgwụ thioctic na-abanye n'ahụ ahụ, ọkwa ya na plasma ọbara ga-adịgide. Tụkwasị na nke ahụ, ụdị iwepụta ngwa ngwa na-enye nnukwu bioavailability nke ngwa ngwa.
Pharmacokinetics nke Tioctacid®
N'ihi ụdị pụrụ iche nke ịhapụ ihe ngwa ngwa, acid alpha-lipoic, nke batara n'ime ahụ n'oge dị mkpirikpi, ruo minit 15-20, na-etinye ya kpamkpam n'ime ọbara site na akụkụ mbụ nke tractestive digestive. N'okwu a, ekwesiri icheta na usoro nhazi nke Thiocacid® BV na ihe oriri na-eme ka ọ ghara ịdị irè nke mkpụrụ ndụ (alpha-lipoic acid). Ịkwado ndụmọdụ ndị dị na ịṅụ ọgwụ - na-ewepu ọkara afọ ọkara otu awa tupu nri - nyere aka gbochie mmekọrịta na-achọghị na nri, n'ọnọdụ a, usoro nke absorption nke mkpụrụ alpha-lipoic acid n'ime ọbara n'oge mmalite nke nri nri ezuola. Ogo kachasị nke tioctic acid na plasma ọbara ruru minit 30 mgbe e weghaara ọgwụ ahụ, ọ bụ 4 μg / ml, ebe mkpụrụ lipoic acid nwere mmetụta "mbụ" site na imeju. Na bioavailability nke mkpụrụ alpha-lipoic acid mgbe ị na-ewere Tioctacid® BV bụ 85%. Ụzọ kachasị mma nke metabolism n'ime ahụ bụ ọnụọgụ na njiko. Ruo 90% nke thioctic acid na ngwaahịa ndị metabolic na-apụ site na akụrụ. Mwepu nke mkpochapu a bụ minit 25.
Na-egosi: polyneuropathy ọrịa shuga na ọrịa shuga
A na-etinye akụrụngwa Thioctic na usoro ọgwụgwọ maka ọrịa ndị na-esonụ: ọrịa nhụjuanya nke metụtara ọrịa na-ejikọta usoro. Radiculopathy. Ọrịa Parkinson. Ogbugbu. Ọrịa ịba ọcha n'anya A na C nke ịdị nwayọọ ma dị oke njọ. Diabetic retinopathy na macular edema.
Nkwekọrịta iji jide Tioctacid®
Ruo taa, enweghi ihe kwesiri ntukwasi obi banyere onodu nke ogwu na aru nke nwanyi n'oge ime ime na umuaka, ya mere, ndi di otua adighi ede Tioctacid. Maka otu ihe kpatara ya, eji ọgwụ maka ọgwụgwọ ndị ọrịa na-erughị afọ 18 adịghị atụ aro. Mmetụta dị iche iche na ọgwụ ndị ahụ bụ ịme ihe.
Ojiji, usoro nke Tioctacid®
Mkpụrụ ọgwụ kwa ụbọchị maka ingestion bụ 600 mg nke ọgwụ (dị na otu mbadamba). A na-ewere ọgwụ ahụ n'ụzọ doro anya na afọ efu, ọkara otu awa tupu ụtụtụ. A na-elo mbadamba ụrọ ahụ dum, n'achọghị afụcha, saa mmiri. Ọ bụrụ na ikpe ahụ dị njọ, Tioctacid® 600T, maka nchịkwa intravenous, na-eji maka ọgwụgwọ. Kwa ụbọchị, onye ọrịa ahụ ji nwayọọ nwayọọ gbanye ya na ọdịnaya nke otu ampoule (600 mg). Ọgwụgwọ ahụ na-adị site na izu abụọ ruo ọnwa, mgbe e mesịrị, onye ọrịa ahụ bufere ọgwụ na Tioctacid® BV. Iji gbochie mmepe nke mmeghachi omume na-achọghị, a ghaghị inye ihe ngwọta na sirinji maka opekempe nke nkeji iri na abụọ.
Ebe ọ bụ na ihe na-arụsi ọrụ ike nke iji ọgwụ ọjọọ eme ihe na-emetụta ìhè, a na-ewepu ampoules n'igbe ahụ tupu a na-edozi ọgwụ ahụ. Mgbe ahụ, a na-ebute ọrịa ahụ na Tioctacid® BV 600 na dose 1 mbadamba kwa ụbọchị.
Mmetụta dị na Tioctacid®
Na akụkụ nke eriri afọ tract na-nchegbu banyere ọgbụgbọ. Ngosipụta ndị ọzọ nke nhụjuanya na akụkụ nke usoro digestive - vomiting, ihe ngbu na ntanwa nke afọ na eriri afọ, izu ike nke stool, mgbanwe na uto - na-enwe ọgba aghara n'ihe ndị dị nnọọ njọ.
Nfụkasị Jeremaya (akpụkpọ itching, rashes na ozu, aṅụ, anaphylactic ujo) adịkarịghị nsogbu.
Site ụjọ usoro nwere ike na-eche banyere dizziness.
General: na nnọọ obere okwu, n'ihi na mmetuta nke glucose mkpofu Filiks nwere ike ịbụ anya mgbaàmà nke hypoglycemia (bịara ikiri ọhụụ, sweating, isi ọwụwa, mgbagwoju anya), nke bụ n'ihi nke ọnụ ke ọbara glucose etoju.
Mmekọrịta ọgwụ ọjọọ na Tioctacid® na ọgwụ ndị ọzọ
Ọ bụrụ na eji ọgwụ ahụ eme ihe na cisplatin, a ga-eme ka mmetụta nke cisplatin pụta.
Ebe ọ bụ na thioctic acid, nke nwere Tioktatsid® BV Tioktatsid® 600T, na-akwalite nkịtị metal adịghị atụ aro n'out oge na ígwè preparations. Oge ime n'etiti Tioctacida® na nkwadebe ígwè, calcium, anwansi kwesịrị ịbụ na ọ dịkarịa ala awa abụọ. N'ọnọdụ ebe a na-eji Tioctacid® mee ihe n'ụzọ na-adaghị adaba na ọgwụ hypoglycemic ora ma ọ bụ insulin, mmetụta nke hypoglycemic nke ndị ọrụ ndị a nwere ike ịkọ ọzọ. Ọ dị mkpa ịhụ ọdịnaya nke glucose n'ọbara, karịsịa na nhazi mbụ nke ọgwụgwọ.
Ntuziaka pụrụ iche
A naghị ekpuchi ọgwụ na ampoules na ọkụ ruo ozugbo eji ya. Maka oge ọgwụgwọ ọ dị mkpa ịhapụ ịṅụ ethanol, ebe ọ bụ na nke ikpeazụ a nwere ike bụrụ ihe na-enye aka na mmepe nke polyneuropathy.
Analogues, price, reviews banyere Tioctacid®
Ọnụahịa nke Tioctacid® n'ụdị ampoules bụ ihe ruru 1500 rubles, n'ụdị mbadamba - 1700-3200 rubles. Ihe nkwakọba kachasị mma bụ 100 mbadamba nkume maka ọnwa atọ.
Tioctacid® bụ naanị ọgwụ dị ugbu a nke nwere ụdị mwepụ ngwa ngwa, bụ nke na-eme ka ọ dịkwuo ụbụrụ nke ahụ na-etinye ya n'ahụ.
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