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"Valium" - bụ ... Description, ntụziaka, edinam ogbo

"Valium" - na ọ bụ n'ihi ọgwụ? Azịza nke ajụjụ a ị ga-ahụ a obere n'ihu. Anyị na-agwa gị banyere otú ngwá ọrụ a na-arụ ọrụ, ihe Njirimara ya e ji dị ka o kwesịrị na ihe-etolite, ọ dị.

The ụdị na mejupụtara nke nkwakọ

"Valium" - a ọgwụ na ike zụrụ n'ụdị ntụtụ, nakwa dị ka mbadamba. Nke ahụ bụ a akụkụ nke ndị a ego?

nwere 5 mg diazepam na 1 ml ngwọta maka ogwu ogbugba. Ndị dị otú ahụ a agwọ ọrịa a na-ahịa ke 50 ma ọ bụ 10 ọchịchịrị iko ampoules of 2 ml, enịm ke katọn.

Banyere mbadamba, ha nwere ike ịnwe 10 ma ọ bụ 5 mg nke diazepam, ma ndị na-esonụ ọzọ Efrata: ọka starch, lactose anhydrous, calcium stearate, pregelatinized starch, e ji esiji ákwà.

Pụtara "Valium" na mbadamba ụdị juru n'ọnụ ke katọn, nke nwere a Valium Valium.

Pharmacology ọgwụ

"Valium" - a ọgwụ na-egosipụta anxiolytic, miorelaksiruyuschee, sedatives, hypnotics na mgbochi ọdịdọ Njirimara.

Tupu anyị na-agwa gị banyere usoro nke ihe nke ego, ọ ga-aghọta na ọ bụ.

Drug "Valium" nwere ndị na-esonụ proprietary aha - "Diazepam". A ọgwụ bụ ìgwè nke benzodiazepines na-enwe oké mkpa na nkà mmụta ọgwụ.

"Valium" - a ọgwụ nke, n'ihi na nke anxiolytic ọrụ, aka esịtidem nchegbu, egwu, nchekasị na nrụgide. Ọkachamara na-ekwu na "Diazepam" dose-dabere utịp ke Central ụjọ usoro. Ndị ọzọ okwu, obere obere (banyere 2-15 mg kwa ụbọchị), nke a ọgwụ ọjọọ na-eme na-akpali akpali mmetụta, na nnukwu (ihe karịrị 15 mg kwa ụbọchị) - ogwuura.

atụmatụ ọgwụ

Gịnị dị ịrịba ama bụ ụzọ dị ka "Valium"? Action (Central muscle relaxant) nke ọgwụ jikọtara a ibelata polysynaptic na-aghọ nkọ na ọgidigi azụ. Ịnata a nkwadebe na-eduga ná a gụnyere ya ná ọbara mgbali, mmụba nke akwara arịa, nakwa dị ka mma iguzogide ọrịa ụbụrụ hypoxia na ihe mgbu ka ukwuu mbata.

kinetics

The agwọ ọrịa "Valium" analogs nke na-egosi n'okpuru, na-etinye obi gị dum na eriri afọ tract (ọnụ). Mgbe a absorption pụtara na 75% na kacha ịta na-ruru mgbe 1.5 awa.

The ndu mgbanwe nke ọgwụ na imeju. N'ụdị a na-arụsi ọrụ ike metabolite na a ọkara ndụ. N'ịhọpụta ọgwụ ka ụmụ ọhụrụ mmetụta ruru mgbe 30 awa, na ndị agadi, na ndị okenye - site 100, na awa 48, karị. Na nke a na ọnụ ọgụgụ imeju pathologies ruo ogologo oge ka 4 ụbọchị.

E lee ya anya nkwadebe ewepụtara ahụ mmadụ tumadi site na akụrụ (90%) n'ụdị conjugates, nakwa dị ka na-agbanweghi agbanwe (2%) na ọnụ na na nsị (8%).

na-agba akaebe

Na ihe ọrịa ọrịa nwere ike na-kenyere a "Valium"? Nyocha ọkachamara na-akọ na a ọgwụ na-egosi na-enweta n'okpuru ndị na-esonụ ọnọdụ:

  • mgbu nke skeletal uru na mpaghara trauma;
  • nchegbu ọrịa;
  • myositis, ogbu na nkwonkwo, bursitis, ọrịa pelvis-spondylitis, adịghị ala ala na-aga n'ihu polyarthritis;
  • tetanus;
  • ọbara mgbali elu, dysphoria, gastric ọnyá afọ na duodenum 12 (ka ihe ndị ọzọ n'aka), myocardial infarction;
  • ehighị ụra nke ọma;
  • rịaworo;
  • spastic ọnọdụ, tinyere ọrịa ụbụrụ, ogbu na nkwonkwo na skeletal muscle erughị ala na athetosis;
  • nsí ọgwụ ọjọọ;
  • vertebral syndrome;
  • mmanya ndọrọ ego syndrome na ngosipụta dị ka nchekasị, ahụ erughị ala, n'ahụhụ, tremor;
  • ọnọdụ epilepticus, ọgwụgwọ nke ọdịdọ;
  • psychosomatic ọrịa na ọrịa ụmụ nwanyị na obstetrics (eg, menopausal na ịhụ nsọ, gestosis, na ikwado oru);
  • eczema na ọrịa ndị ọzọ na-ebu itching na ogwe;
  • Meniere ọrịa ;
  • hallucinatory-paranoid ala, moto excitation nke dị iche iche si malite (na ọrịa uche na neurology);
  • general ná Nkụnwụ na premedication (eg, tupu ịwa ahụ na endoscopic usoro).

contraindications

Mgbe ị na-ekwesịghị iji nke a ọgwụ ọjọọ dị ka "Valium"? Mmetụta nke a ọgwụ abụghị otu dị ka anyị ga-achọ, ọ bụrụ na ị na-anabata ya:

  • na hypersensitivity;
  • Coma, ujo;
  • nnukwu mmanya igbu egbu;
  • nnukwu iche nke ọrịa imeju;
  • myasthenia gravis;
  • n'akuku-mmechi glaucoma;
  • na ụmụ obere karịa 6 ọnwa;
  • n'oge lactation, na nke mbụ trimester nke afọ ime.

Ọgwụ "Valium": ntuziaka maka ojiji

Kenye atụle a n'aka ga-enwe nanị ahụmahụ ọkachamara. N'ihi na okenye ọrịa a dose nke ọgwụ mgbe onu ochichi kwesịrị 5-20 mg kwa ụbọchị. Nke a buru ibu nke ọgwụ kpebisiri ike dabere na ogo nke ọrịa mgbaàmà, nakwa dị ka ngụkọta adakarị picture.

The kacha ekwe omume dose ọgwụgwọ bụghị ihe karịrị 10 mg. ọgwụ N'ezie, nke a pụtara na ihe banyere nchegbu ọrịa ga-adịru banyere 6 izu. Mgbe oge a ga-ezo aka ịga dọkịta, nke mere na ọ were a kacha nta mmezi onunu ogwu.

-Ekpochapụ nke ọgwụ nke nta nke nta na-ewere.

Na mberede mgbe, ifịk agwọ ọrịa ka ga-ndinọ parenterally (intramuscularly ma ọ bụ intravenously). Na nke a, a dose of 2-20 mg.

Na igba ogwu n'akwara infusion nke ọgwụ ga-ndinọ nwayọọ nwayọọ, na a ọnụego adịghị nnọọ 0.5-1 ml kwa nkeji.

mmetụta

Dị ka ọgwụ ọ bụla, na-ewere na-atụle ọgwụ nwere ike ime ka ihe oghom mmeghachi omume. Ndị a gụnyere ndị na-esonụ:

  • bradycardia ma ọ bụ hypotension;
  • ebelata ịta na mmeghachi omume ọnụego;
  • riri ahụ ọgwụ ọjọọ;
  • dizziness na isi ọwụwa;
  • mmepe nke paradoxical Jeremaya mere, nke nchegbu, ehighi ura, ịmụ anya arọ nrọ, na ihe ọdịdọ;
  • ebe nchekwa impairment (obere);
  • n'akụkụ Jeremaya mere na-agbanye saịtị;
  • ije ọrịa ndị dị otú dị ka dysarthria na ataxia;
  • mmebi nke akụrụ na imeju, gootu atony, ebelata libido na potency (ogologo oge nke ọgwụ);
  • nfụkasị Jeremaya;
  • ndọrọ ego syndrome;
  • ebelata arụmọrụ, na ike ahu ike.

Ná nhọpụta nke ọgwụ na-enwe ndidi ọ dị ezigbo mkpa na-agwa ya na nke a bụ a ọgwụ. Mgbe na-ewere a mara psychotropic gị n'ụlọnga mgbanwụ, nke nwere ọtụtụ oghom mmetụta, otu nke karịsịa natara eri ahụ na ndọrọ ego.

Dr. e a na nkà mmụta ọgwụ na iwu ji na-agwa ndị ọrịa banyere omume oghom mmetụta nke ọgwụ na ahụ ya, dị ka nke ọma dị ka na-enye ndị ọzọ ọgwụgwọ nhọrọ.

ovadozu nke na nkà mmụta ọgwụ

Overdosing atụle wetara n'aka esonyere ndị dị otú ahụ ihe mgbaàmà dị ka CNS ịda mbà n'obi. A yiri onu nwere ike ná mgbanwe nke ogo, sitere na site iro ụra na-agwụcha amaghị onwe ya. Ọzọkwa, mgbe na-ewere elu doses nke ọgwụ na onye ọrịa ahụ na o kwere omume hypotension, mgbagwoju anya na akụkụ okuku ume na ịda mbà n'obi.

The ọgwụgwọ nke ọnọdụ ndị dị otú na proviso, ma ọ bụrụ na onye ọrịa bụ adịghị, na-agụnye itinye n'ọkwa nke emesis na ojiji nke ọrụ carbon. Na ikpe, ma ọ bụrụ na onye ọrịa bụ amaghị ihe ọ bụla, ọ na-na-asa site na a na afo nyocha, nakwa dị ka symptomatic ọgwụ, screening mkpa ọrụ ma na iwebata ọmụmụ aka diuresis.

Ijide oké n'ahụhụ onye ọrịa, i nwere ike na-ekenye ya barbiturates.

Mmekọrịta ọzọ ike n'aka

The agwọ ọrịa "Valium" akpata potentiation mmanya mmetụta, hypnotics, anticonvulsants, hypotensive elekọta mmadụ na Antihistamines, na antipsychotics, n'ozuzu ọgwụ na-akụnwụ, tricyclic antidepressants, muscle relaxants na analgesics.

Analeptic stimulants na ike budata belata ọrụ "Diazepam" ọgwụ ọjọọ.

Antacids ibelata ọnụego, ma ọ bụghị na ọkwa nke absorption nke ọgwụ.

Dị otú ahụ inhibitors nke microsomal ọxịdashọn dị ka "Cimetidine", "Omeprazole" "ketoconazole" "fluoxetine" na "Fluvoxamine" ịgbanwe pharmacokinetics nke ọgwụ n'okpuru echiche, na-amụbakwa oge nke ya na-adakarị mmetụta.

"Rifampicin" ebelata ịta nke "Diazepam" na ọbara, na "Erythromycin" slows ala ya metabolism na imeju.

yiri ọgwụ ọjọọ

Gịnị nwere ike dochie a ọgwụ dị ka "Valium"? Analogues na Russia na-adịghị ere pharmacies. Ọzọkwa, ọgwụ ndị a na-tọhapụrụ nanị mgbe ngosi nke ọgwụ na ahụ ike ọgwụ.

Dochie ọgwụ nwere ike "sibazon", "diazepam" ma ọ bụ "Diapamom". Otú ọ dị, nke a ga-eme nanị mgbe oge na dọkịta.

The na-eri nke ọgwụ

Dị ka m kwuru n'elu, ịzụta ọgwụ ọjọọ, "Valium Roche" na Russia nwere ike ọ bụghị na ọ bụla ahịa ọgwụ. The na-eri nke ọgwụ - banyere otu puku rubles (kwa mkpọ).

The price ego na UK na ndị ọzọ na mba Europe, na-emekarị ihe abụọ na narị abụọ na iri ise na pound kwa puku mbadamba (10 mg).

Ịzụta na obodo ahụ bụ ndị dị otú ahụ a ọgwụ ga-ezute niile chọrọ nke nchekwa na àgwà, ndị ọkachamara nwere ike ikwu na itinye ndabere, ebe ị ga-nyere ihe ọmụma zuru ezu banyere ya nnweta na pharmacies na kasị uru ahịa.

Consumer reviews banyere ọgwụ

"Valium" - ọ bụ nnọọ ihe na-ewu ewu n'etiti ndị ọrịa a ọgwụ nke na-eji dị ka ihe anxiolytic, miorelaksiruyuschego, sedatives, hypnotics, na anticonvulsants. Dị ka nzaghachi ọtụtụ ndị na-eji ọkụ, a na-ewere ukwuu irè ọgwụ maka ọrịa dị iche iche, gụnyere Akwụkwụ na-adọ, nsogbu ihi ụra, nchegbu na na. Ọzọkwa na-ewere ya na-enyere aka mfe mgbaàmà dị ka n'ahụhụ, tremor na iwepụ ịmụ anya arọ nrọ.

Otú ọ dị, e nweghị ndị dị otú ahụ ngwá ọrụ na-ga-asatọ onye ọ bụla. Ụfọdụ ndị na-eji a ọgwụ adịghị enwe obi ụtọ. Ha mara na ọgwụ na-amalite na-eme ihe nanị mgbe a izu. Ke adianade do, na nọgide were agwọ ọrịa na-akpata a ọnụ ọgụgụ buru ibu nke n'akụkụ Jeremaya mere na-eduga ná riri ahụ.

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