Ahụ ike, Preparations
"Artrokol" (jel): ntuziaka maka ojiji, analogs na reviews
Olee otú m ga-eji ọgwụ ọjọọ, "Artrokol" (jel)? Ntuziaka maka ojiji nke ọgwụ ga-kọwara n'isiokwu a. Ọzọkwa, ị ga-amụta ihe site n'ihe ọgwụ kenyere ọrịa, ma o nwere analogues, na ihe ọ bụla kwuru banyere ya doo n'ji.
Formulations, nkwakọ ọgwụ ọjọọ na ya udi
"Artrokol '- jel (2.5%) maka mpụga were. Na ire ọ ga-abịa na aluminum tube 45 dịkwa na a kaadiboodu igbe ọnụ na ịṅụ ọgwụ bụ a mpempe akwụkwọ na zuru ezu ntuziaka maka ojiji.
Na e dere mpụga ọgwụ "Artrokol" (jel)? 100 g nke a na-ajụ nwere 2,5 g nke nọ n'ọrụ mgwa, dị ka ketoprofen. Ke adianade do, na ọgwụ a na-atụle na-agụnye ndị na-esonụ support ọcha: trolamine, Carbomer 980, 96% ethanol, ọcha mmiri na methyl parahydroxybenzoate.
Ụkpụrụ nke ime ihe nke a agwọ ọrịa
"Artrokol" - a jel, na-arụsi ọrụ ike mgwa na-ketoprofen. Sị na agwọ ọrịa nke na ìgwè nke ndị so ná ndị mgbochi mkpali ọgwụ ọjọọ, dị ka nke ọma dị ka nkwekọrịta nke arylpropionic acid.
Base ihe onwunwe na-ewere agwọ ọrịa na-enye mgbochi mkpali na analgesic mmetụta, nke pụtara n'oge na-abụghị nhọrọ mgbochi nke Cox-1, bradykinin na Cox-2, na akpụkpọ ahụ stabilization (lysosomal) na mgbochi nke macrophage Mbugharị.
Ke adianade do, ọgwụ ọjọọ, "Artrokol" (jel) egosipụta mgbochi mkpali na ahu izizi Njirimara. Ọ bụ ike na-eme ihe na n'oge na mbubreyo cell vaskụla adọ nke aza. Ọzọkwa, a ọgwụ slows ala platelet aggregation.
The pharmacokinetic e ji mara
Dị ka mmasị ntuziaka, ketoprofen (n'ọrụ mgwa nke agwọ ọrịa) mgbe Nde ngwa ka akpụkpọ etinye obi gị dum, na mgbe penetrates n'ime etiti nke mkpali usoro na n'oge a ogologo oge na-ekwusi chọrọ ọgwụgwọ ịta na arọ.
Absorption nke ọgwụ n'ime systemic mgbasa bụ ntakiri (banyere 5% nke dose eji). Na nke a, na absorption n'ime ọbara stream bụ nnọọ ngwa ngwa.
Ịta nke nọ n'ọrụ mgwa nke ọgwụ (iji 50-150 mg nke ketoprofen) na ọbara mgbe 7.5 awa bụ naanị 0.08-0.15 mg / ml.
Drug "Artrokol" (jel) na nzube ya?
The egosi maka ojiji nke jel n'okpuru echiche na-na-esonụ na-ekwu:
- myalgia, rheumatic na rheumatic si;
- ọrịa nke nweekwa usoro (gụnyere ọrịa ogbu ogbu na nkwonkwo, articular syndrome n'oge exacerbation gout, ankylosing spondylitis, psoriatic ogbu na nkwonkwo, osteochondrosis, osteoarthritis nke dị iche iche orunótu, mgbu lesion nke akwara, ụdọ, sciatica, bursitis ma ọ bụ ọrịa azụ mgbu);
- akụkụ nke mgbagwoju ọgwụgwọ nke mkpali pathologies veins (e.g., phlebitis, periphlebitis), Lymph ma ọ bụ Lymph arịa (e.g., lymphangitis, elu elu lymphadenitis);
- post-traumatic mbufụt nke nweekwa usoro na adụ anụ ahụ (gụnyere symptomatic ọgwụgwọ nke na-adịghị mgbagwoju unan, gụnyere sprains, egwuregwu unan, sprains ma ọ bụ anya mmiri nke akwara na akwara njikọ, bruises, post-traumatic mgbu).
Bans ojiji nke
Gịnị ka "Artrokol" ude na-enyere aka, anyị na-akọwara n'elu. Otú ọ dị, nke a pụtara na e nwere contraindications. Ndị a gụnyere ndị na-esonụ:
- afọ n'okpuru 12 afọ;
- elu uche na ndị ọcha nke ọgwụ nakwa dị ka acetylsalicylic acid ndị ọzọ NSAIDs;
- nke-atọ trimester nke afọ ime na ara.
Drug "Artrokol" (jel): ntuziaka maka ojiji
Maka ọgwụgwọ nke jel iyipu 5.4 cm ogologo n'okpuru echiche pụtara etinyere ndị ahụ na-chọrọ ebe adụ rubbing massaging mmegharị ruo mgbe ya zuru absorption.
Ọ ga-kwuru na ibu ebe nke otụk ebe, ọzọ ọgwụ na-aga n'ime a ọgwụ na usoro. N'ihi ya pyatisantimetrovym warara agwọ ọrịa "Artrokol" kwekọrọ na 100 g ketoprfena.
Mgbe ude a na-eji, ọ ga-ozugbo na-asa aka.
E lee ya anya jel na-ekwe na-eji na njikọ na ndị ọzọ ka ọgwụgwọ nwere a ketoprofen (e.g., na njikọ na mbadamba, capsules, rectal suppositories).
The kacha dose of gị n'ụlọnga bụ 200 mg kwa ụbọchị. Nke a bụ ego nke ọgwụ adịghị adabere n'ụdị ọgwụ.
Na oge nke ọgwụgwọ N'ezie kwesịrị ikpebisi ike n'otu n'otu site na ịga dibịa. Otú ọ dị, ọ ga-kwuru na ihe liniment n'ihi na ihe karịrị 10 ụbọchị a n'usoro ajuru aju.
Ekwe Omume mmetụta
Gịnị mmetụta ọjọọ nwere ike ime ka ọgwụ "Artrokol" (jel)? Ntụziaka kwuru banyere ndị na-esonụ mmetụta ọjọọ nke ọdịdị:
- bronchospasm, angioedema;
- asthmatic ọgụ, anaphylactic Jeremaya mere gụnyere ujo;
- nācha ọbara-ọbara, itching, ọkụ ọkụ, ọkụ na ọzịza nke anụ;
- bullous phlyctenular eczema na ike nke na-agbasa ndị ọzọ ebe na iji nweta generalized;
- photosensitivity, bullous ma ọ bụ kọntaktị dermatitis;
- ọgbụgbọ, Stevens-Johnson syndrome, vomiting;
- agba ọbara, afo ọnyá, afọ ọsịsa, nrekasi obi, afọ ntachi;
- Aghara nke akụrụ ọrụ, exacerbation nke gbasara akụrụ odida na-adịghị ala uwa, interstitial nephritis na gbasara akụrụ odida.
Ọ kwesịkwara kwuru na mgbe eji jel "Artrokol" nwere ike ime ka ndị ọzọ n'akụkụ Jeremaya mere na site digestive usoro na urinary usoro. Siri nke mmetụta ndị a na-adabere na ego nke ọgwụ ọjọọ na permeation ike nke ya nọ n'ọrụ mgwa, mesoo ebe size, ọnụego na oge nke ọgwụgwọ ọnọdụ nke anụ.
Anyị nwere ike ikwu na ndị agadi na-adịghị ike na oghom mmetụta nke NSAIDs na ọgwụgwọ.
N'oge ime na lactation
Enwere m ike iji ọgwụ "Artrokol" (jel) n'oge ime na ara? Na N'ezie nke nwere na òké, ọ hụrụ na nke ego na-adịghị eme ka teratogenic na embryotoxic mmetụta na-eto eto ụmụ anụmanụ. Otú ọ dị, ọ ga-ahụ kwuru a obere embryotoxic mmetụta ka a hụworo nwere na rabbits.
Ebe ọ bụ na nchekwa nke ketoprofen na ụmụ nwaanyị dị ime na a na-akwado site ọ bụla ọmụmụ, ndị ọkachamara na adịghị ike ikwu iji ngwá ọrụ a na-abụ nne.
Ọzọkwa, ọ ga-ahụ kwuru na ketoprofen na ndị ọzọ na inhibitors nke prostaglandin njikọ pụrụ ịkpasu gbasara akụrụ toxicity, akpa ume na gbasara obi usoro nke nwa ebu n'afọ.
The ire ere ngwaahịa nke ego na-hụrụ na mmiri ara. N'ihi nke a, jel "Artrokol" kwesịghị ndinọ na nwa ara na-nwanyi.
kpọmkwem ozi
Nkwadebe "Artrokol" (jel), nke analogs e depụtara n'okpuru ebe, ọ na-aju itinye akpụkpọ ebe enweghị nchịkwa mgbanwe ndị dị otú ahụ dị ka ihe otutu ma ọ bụ eczema. The otu na-emetụta nje ebe ma ọ bụ na-emeghe ọnyá.
Ị ga-zere ọgwụ na kọntaktị na mucous membranes. Mgbe iji ọgwụ ga-akwọ aka.
Nke a na ngwá ọrụ bụ kwesịrị ekwesị maka na occlusive dressings.
N'oge ọgwụgwọ "Artrokolom" na izu abụọ mgbe omume, ọ bụ na-achọsi ike iji zere kọntaktị na akpụkpọ kpọmkwem ìhè anyanwụ.
"Artrokol" (jel): reviews na yiri preparations
Site analogues nke a ọgwụ na-agụnye ọgwụ ndị dị otú ahụ dị ka "Karmolis-jel", "Indomethacin", "diclofenac", "Remisid", "Vipratoks", "Denebola", "Nzube nke T", "chondro ike", "Ibuprofen" "Ketonal" na ndị ọzọ.
Ihe ndị mmadụ na-ekwu banyere ọgwụ ọrụ? Ha kọrọ na jel "Artrokol" na-anọchi anya ihe irè mgbochi mkpali n'ụlọnga. Ọ na-emeso nke ọma ndị enweghị nchịkwa ọnọdụ dị ka myalgia, ọrịa nke locomotor usoro, mkpali oria nke veins, post-traumatic mbufụt.
The ọghọm nke a ọgwụ maka mpụga na ngwa na-agụnye a plurality nke n'akụkụ-mmetụta nke egosipụta onwe ha mgbe were jel. Ọtụtụ mgbe, ndị ọrịa na-hụrụ nācha ọbara-ọbara, itching, aṅụ, ọkụ na ọzịza nke anụ ahụ, dị ka nke ọma dị ka ọgbụgbọ, eczema, afo ọnyá, afọ ọsịsa na nrekasi obi. Ọzọ mwepu nke na-ewere ọgwụ ọjọọ bụ na ọ na-apụghị kenyere ka ụmụ nwaanyị dị ime, nakwa dị ka eji n'oge lactation.
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