Ahụ ikePreparations

Drug 'Atenolol Nycomed'

N'ihi na ọgwụ ọjọọ, "Atenolol Nycomed" e chemical, na mba mgbochiume na aha "Atenolol". Na asụsụ nke chemists pharmacologists structurally ọgwụ na-egosi dị ka (RS) -4- (2-hydroxy -3- (isopropylamino) phenyl-acetamide. Mbadamba "Atenolol" na-anọchi anya oboevypuklye ntekwasa mkpụrụ ọgwụ nke na-acha ọcha na agba, nwere a Capsule udi. Isi ahụ na-nyere notch maka a ezumike na otu aka, e nwere ihe ịrịba ama AV55 na AV57.

Na otu mbadamba, dabere na ntọhapụ ụdị nwere ike ịnwe na iri ise ma ọ bụ otu narị milligrams nke atenolol. Inyeaka mmiri eji talc, gelatin, propylene glycol, titanium dioxide, magnesium stearate, ipromeloza 2910 (15sP), ọka starch, sodium lauryl sulfate, arọ magnesium carbonate.

Medicine "Atenolol Nycomed" omume dị ka a beta1-nhọrọ (cardioselective) adrenoceptor igbochi gị n'ụlọnga, akpụkpọ ahụ kwụsie ike ọrụ bụghị. Ngwá ọrụ a na-egosi antianginal, antiarrhythmic na hypotensive mmetụta. Ọ bụ ike nke na igbochi beta-adrenergic anabata nke obi, na-ebelata myocardial mmetuta nke obi ebere nkewa autonomic ụjọ usoro na catecholamines, nke igbasa na ọbara. Medicine "Atenolol" mmetụta na mbenata imi automaticity, apụta na obi ọnụego ka a akwụsị na n'oge omumu. Nke a stabilizes usoro na excitation nke myocardial contractility, ibelata mmetụta AV-conduction. Na ya ngwa e nwere a ọnụ ke myocardial oxygen ina. Mma na-emetụta ndị Ịhazi ojiji ọgwụ "Atenolol" na ẹsụhọde ọbara mgbali. Stabilization nke antihypertensive mmetụta emee site na njedebe nke abụọ n'izu nke n'ikuku.

Nkwadebe "Atenolol Nycomed" n'elu onu n'ikuku usoro ike etinye obi gị dum na digestive tract na olu nke 50-60% nke ndinọ dose. Anyụpụ na mmamịrị na a ọkara ndụ-nke 6-7 awa. A oge na ọrịa na gbasara akụrụ impairment, dabere na ọnụego nke glomerular filtration.

Egosi maka ọgwụ bụ "Atenolol Nycomed" nwere ụdị nke ọbara mgbali na tachyarrhythmias (gụnyere imi). Mee ọgwụ na dị ka a mgbochi gị n'ụlọnga maka rịaworo ọgụ.

The kwa onunu ogwu nke ọgwụ n'ihi na ndị okenye na ọgwụgwọ nke rịaworo na ọbara mgbali esịmde 50-100 mg. Admission mbadamba mere ruo ugboro abụọ n'ụbọchị anya nke eziokwu ahụ bụ na kwa ụbọchị dose ekwesịghị gafere 200 mg. Iji na-asa ala ọgwụ kwesịrị a obere ego mmiri.

The na nkà mmụta ọgwụ na-eji na na nlezianya dị na-atụ aro nke ịga dibịa. Self-ọgwụ na-adịghị ekwe. Ọgwụ "Atenolol Nycomed" nwere mmetụta. The obi usoro nwere ike ikwu ọdịdị bradycardia, AV-conduction disturbances, ị pụrụ inweta sensations nke paresthesia na oyi na-atụ aka na ụkwụ, na ụfọdụ na-apụta ìhè mgbaàmà nke obi ọdịda. Digestive tract mkpatụ ezighị-ọgwụ ọgbụgbọ, afọ ntachi, afọ ọsịsa, akọrọ ọnụ (obere), na endocrine usoro - ekwe omume mmepe nke a hypoglycemic ọnọdụ na ọrịa na-ata ahụhụ si na-arịa ọrịa shuga, urogenital usoro - ekwe omume ọnụ ke potency. CNS oghom Jeremaya mere nwere ike na-egosipụta na isi ọwụwa, dizziness, nsogbu ihi ụra, ịda mbà n'obi, mmetụta nke ike ọgwụgwụ. Ọ dịkwa ike nfụkasị Jeremaya, itching, na nācha ọbara-ọbara. Ikpe amplification igba ajirija, Mbelata adọka ọmụmụ secretion e dere, omume nke conjunctivitis.

Ọzọkwa, e nwere ọtụtụ ihe ndị contraindications. Na ha ndepụta gụnyere onye nkebi nke-adịghị ala ala obi ọdịda, bradycardia, hypotension, ubara uche ọgwụ, na ndị ọzọ.

Nọgidenụ na-ahụ ọgwụ na a kpọrọ nkụ, na-echebe site ìhè, na mwepu nke ụmụ. Ụlọ okpomọkụ na 25 Celsius C. A ọgwụ na-ekwusi ya Njirimara nke afọ ise.

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