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Ọgwụ "Sulpiride": reviews, na-egosi, analogs

Psychosis ná mgbanwe nke ogo so ndi mmadu mgbe. N'ime ọtụtụ narị afọ e kweere na nwere site ekwensu na a na-arịa ọrịa madu, ya mere "ihe ngwọta" nsogbu a kemgbe kwesịrị ekwesị. Tupu e kere eke nke neuroleptic ọgwụ enyemaka nsogbu uche emepụta herbal agwọ ọrịa mepụtara na ndabere nke belladonna, henbane, opiates. Mere ka ọgwụgwọ na calcium (igba ogwu n'akwara) na n'imikpu onye ọrịa na a na-ehi ụra ọgwụ.

The nnọọ mbụ antipsychotic chlorpromazine nwere ike na-akpọ, bụ nke e ifịk ifịk na-eji maka ọgwụgwọ nke ọrịa na iche echiche ike nsogbu ebe ọ bụ na 1953. Ugbu a, ndị ndepụta antipsychotic ọgwụ, antipsychotics budata gbasaa. Otu nke ọtụtụ-eji ọgwụ ọjọọ nke otu a bụ "Sulpiride". Nleba akọwa ya dị ka a ukwuu gbara gharịị antipsychotic.

pharmacodynamics nke ọgwụ

Neuroleptic mmetụta "sulpiride" antidofaminergicheskim metụtara na-eme ihe, m. E. Na Central ụjọ usoro ọgwụ nkanka tumadi dopaminergic anabata. Dopamine bụ ihe dị mkpa akụrụngwa nke "ụgwọ ọrụ usoro" nke ụbụrụ - akpali ụtọ sensashion, na-eju afọ karịa, n'aka nke ya, na-emetụta ndị mmụta ma motivational Filiks. Na elu nke ọma doses, na-emepụta na usoro nke ọ bụla nti ahụmahụ (na nke onye uche nke a onye) - n'ikuku nke na-atọ ụtọ nri, na-enwe mmekọahụ, ọ dịghị obi ụtọ aru sensations. Na-amụba ego nke dopamine na Central ụjọ usoro na-akakwa mma psychological nkasi obi, na a ọnụ - ịzụlite mgbaàmà nke ịda mbà n'obi.

Action "sulpiride" na a dose uku 600 mg (kwa ụbọchị ego nke ọgwụ) bụ antipsychotic okike. Ọ bụrụ na ndị Dosages na-erughị 600 mg - ọzọ juru ebe niile stimulant na antidepressant mmetụta. Otú ọ dị serotonicheskie, histamine, adrenergic anabata ọgwụ nwere obere mmetụta.

Ọgwụ - analogues

The agwọ ọrịa "Sulpiride" - gbara gharịị neuroleptic, bụ ìgwè nke nnọchianya benzamides - nwere a zuru ezu ọnụ ọgụgụ buru ibu nke ọgwụ ndị yiri na mejupụtara na nwere mmetụta. E nwere ọgwụ ọjọọ nke dakọtara na koodu ATC 4th larịị. Ndị a bụ ndị "Betamax", "tiaprid", "Eglonil". E wezụga ndị a, a sara mbara n'ji ina "Prosulpin", "Eglek" "edinem" "Vero Sulpiride", "Sulpiride Belupo." Nyocha nke niile ọgwụ site na-eji ọkụ nwere ike ma ndị nke ọma direction na-adịghị mma. Ọ niile na-adabere na ogo nke ọrịa steeti ahụ ike, ya uche na isi na-arụsi ọrụ ike mgwa - sulpiride, na onunu ogwu nke ọgwụ kenyere na-enweta a dọkịta.

Egosi na-enweta ọgwụ

Sam neuroleptic "Sulpiride", ya analogs nwere a pụtara sara mbara nọ nke mmetụta na ike ga-kenyere na-enweta a zuru ezu oké njọ nke ọrịa. Were ya na ọnụnọ nke isi mgbaka na nnukwu nkebi, na mgbe bụ ala ala. Sulpiridsoderzhaschih n'onye ezi omume ojiji nke antipsychotics n'oge nnukwu ogbo nke mmepe nke delirium (a echiche-aghasa nke okike, Bilie a nsogbu nke nsụhọ sitere na site dizziness na ọbụna amaghị onwe). Ọtụtụ mgbe ọgwụ na-kenyere iche iche koro ndị mmadụ n'elu ọrịa na ịda mbà n'obi, n'agbanyeghị na ha si malite.

Mgbe vertigo nke dị iche iche si malite tụrụ aro na-ewere "Sulpiride" ntụziaka ntuziaka. Nyocha nke ọrịa na n'ụlọ ọgwụ na-ọma e ji mara agwọ ọrịa n'ịgwọ vestibular neuritis, mgbe ọdịda vertebrobasilar-basilar ụdị na otitis media na cranial mkpasasị uche, na Meniere ọrịa (ụba olu nke ọmụmụ na n'ime ntị uji eze, nke na-ewepụta nsogbu na mkpụrụ ndụ maka ịnọgide na-enwe ịha ahu na ya nghazi ohere).

Dị ka a "Sulpiride" akụkụ nke a sara mbara ọgwụ ike ga-eji na ọgwụgwọ eme maka peptic ọnyá afọ ọrịa na agbakasị bowel syndrome.

Ònye kwesịrị izere ịdị na antipsychotic ọgwụ ọjọọ na ndabere nke sulpiride?

Neuroleptics "Sulpiride" ọgwụ analogues nke isi n'ọrụ mgwa nwere a kpọmkwem ndepụta contraindications. Ejila ya ndị mmadụ na hypersensitivity ka sulpiridu na-ata ahụhụ site hyperprolactinemia (budata elu etoju nke hormone prolactin n'ime ọbara). Ntem, a ọgwụ na-adịghị kenyere prolactin-ndabere etuto ahụ (ara cancer, prolactinoma pituitary gland , wdg).

Ọzọkwa, "Sulpiride" (egosi akọwara n'elu) machibidoro ntụziaka pheochromocytoma (hormonally ifịk chromaffin cell etuto ahụ), manic psychosis dị iche iche affective ọrịa na akparamàgwà awakpo Akwụkwụ na-adọ. Unu na-eji nke a ọgwụ sulpiridsoderzhaschih megide backdrop nke nnukwu mmanya igbu egbu, nsí na hypnotic ọgwụ na narcotic analgesics.

Adịghị bụ ojiji nke neuroleptic "Sulpiride" ọrịa noo n'okpuru 18 afọ na ndị inyom n'oge lactation.

Ekwe Omume mmetụta nke

Oghom Jeremaya mere ka neuroleptic onwe ya na analogues "sulpiride" ndidi testimonials na ndị ọkachamara ahụ ike mara dị ka zuru ezu dị oké njọ, budata na-akawanye njọ ọnọdụ nke ndị ọrịa. E nwere a-ekwe omume nke hyperprolactinemia na a dịgasị iche iche nke iche (gynecomastia, dysmenorrhea, frigidity, belata potency, galactorrhea, na-abawanye na ahu arọ).

Ọzọkwa omume ngosipụta nke extrapyramidal syndrome, nke na-egosipụta site enweghị nchịkwa ọrịa nke ukwu na àgwà nke n'amaghi ije emepụta site skeletal mọzụlụ, ịgbanwe na Akwara ụda. Otú ọ dị, mkpọnwụ bụghị a mgbaàmà na-egosi eziokwu nke na extrapyramidal syndrome.

Dị ka n'akụkụ Jeremaya mere ka "Sulpiride" analogs neuroleptic, nwere ike ime tremor, akathisia (enweghi ike ibu na-ezu ike), dyskinesia, ehighi ura, iro ụra, nchegbu elu excitability, ahụ mgbakasị. Pụrụ igosipụta mgbaàmà nke neuroleptic ajọ syndrome, ji autonomic abnormalities, icha mmirimmiri anụ ahụ, hyperthermia.

Mmetụta si eriri afọ tract nwere ike a sensashion nke nkụ ke inua, mmepe nke nrekasi obi, ọgbụgbọ anya, retching, afọ ntachi. Ekwe Omume ebighị nke hepatic transaminases na alkaline phosphatase.

Obi usoro ngwa "sulpiride" nwere ike ikwu na-abawanye na ọbara mgbali (adịkarịghị - a ọnụ ke ọbara mgbali, dizziness), mụbara obi ọnụego, mụbara QT-nkeji. Nnọọ adịkarịghị, ma i nwere ike ịnụ na na "Sulpiride" ọgwụ omume na dọkịta na-egosi na mmepe torsadedepointes ụdị arrhythmia.

Anabata ngosipụta ndị dị otú ahụ dị ka akpụkpọ ọkụ ọkụ, pruritus, eczematous ọnya. Mgbe ụfọdụ, i nwere ike ịnụ banyere ndị mebiri nke visual acuity.

dosing na ngwa circuit mode

Dị ka ntụziaka maka ojiji nke agwọ ọrịa, a na okenye ọrịa dabere na ọrịa kenyere dose of 100-300 mg kwa ụbọchị (kewara 2-3 doses). Oral ngwọta ndinọ dị iche iche onunu ogwu: 100-800 mg kwa ụbọchị maka intramuscular ochichi (tupu ojiji bụchaghị jijiji). The kacha anabata dose maka na onye toro eto bụ 1.6 g

Ọ bụrụ na ọ dị mkpa na-ekenye "sulpiride" ka ụmụ n'okpuru afọ 18, na onunu ogwu ga-gbakọọ na-ewere n'ime akaụntụ arọ na ndabere nke 5 mg kwa kilogram nke ahu aro.

Ọ bụrụ na onye ọrịa nwere a ọnọdụ nke psychosis na nnukwu ma ọ bụ ala ala ogbo, ọgwụ a na-amalite na intramuscular ochichi (400-800 mg kwa ụbọchị). N'ọnọdụ ka ukwuu, oge nke ọgwụgwọ ọ dịkarịa ala izu 2. Ozugbo ahụ ike onye ọrịa, site intramuscular injection zigara n'ikuku "sulpiride" n'ime a Erere. Neuroleptic "Sulpiride" ndidi reviews-akọwa dị ka dị irè ọgwụ. Duration nke N'ezie nke ọgwụ nwere ike kpebisie ma gbanwee naanị site ịga dibịa.

oké doses

Ọ bụla kpọmkwem mgbaàmà na-egosi eziokwu nke uku karịa ime doses n'elu, ọ dịghị. Na-emekarị na ọnọdụ ndị a, e nwere ubara ọbara mgbali, bịara ikiri ọhụụ. Ikekwe mmepe nke ogwuura (suppression nke nsụhọ iwe na ọgwụ ọjọọ, obi mmetụta, mgbe elu doses - hypnotic). N'ọnọdụ ka ukwuu, mmetụta nke ọgwụ "Sulpiride" ndidi testimonials egosi ọdịdị ọgbụgbọ, akọrọ ọnụ, mụbara sweating, vomiting. Na obere okwu ịzụlite extrapyramidal mgbaàmà, gynecomastia nwere ike ime nwoke ọrịa (ara ịmụba ọnụ ọgụgụ). Nnọọ adịkarịghị ekwu okwu nke akpọ parkinsonism, amaghị onwe ya.

Dị ka nhọrọ ngwọta maka "sulpiride" offline, symptomatic omume na-atụ aro, dabere na ọnọdụ nke onye ọrịa. Mgbe ụfọdụ, tinye holinoblokatory Central edinam.

On ihe ntị?

Nnọọ niile ngwaahịa antipsychotic otu (gụnyere sulpiridsoderzhatsie "Betamax", "Vero Sulpiride", "Prosulpin", "Sulperid Belupo", "Eglonil", "Sulpiride") reviews ọkachamara na-arụ ọrụ ntuziaka na machibidoro ndabere nke mmanya na-aba n'anya. N'ihi na ọrịa na Akwụkwụ na-adọ na-atụ aro na-eduzi na-adakarị na electrophysiological ọmụmụ e sulpiride ọ lowers fọrọ maka ọdịdọ ọrụ. Ọ bụrụ na ọgwụ a na-eji concomitantly na ọgwụ ọjọọ na-amụba ihe ize ndụ nke ventricular arrhythmias, dị ọrịa na-achọ mgbe nile nlekota nke ngwá. Mụbara QT-nkeji na-adabere na dose.

Ọ bụrụ na n'oge ọgwụgwọ, "sulpiride" ndị mgbaàmà nke hyperthermia (a eziokwu na-arụtụ aka na mmepe nke neuroleptic ajọ syndrome), site n'iji ọgwụ ga-kwụsịrị.

Mberede cessation nke ọgwụ "sulpiride" pụrụ ịkpasu ndọrọ ego mgbaàmà. Maltitol bụ ugbu a na ọgwụ na-eme ka ọ gaghị ekwe omume iji ndị mmadụ na-ata ahụhụ site na fructose ekweghị ibe nọrọ.

N'oge dum ọgwụgwọ oge kwesịrị-nọgide na ugbo ala na mmejuputa management arụmọrụ-achọ ngwa ngwa omume psychomotor na elu ịta.

Sulpiridsoderzhaschie ọgwụ na ime

Women n'oge ime "Sulpiride 'reviews ekpe na ihe ndị kasị mma direction. Oke allowable dose ka nwanyị dị ime bụ 200 mg kwa ụbọchị na-akpasu teratogenic mmetụta (nupụsịrị nke ẹmbrayo development). The dịtụ ukwuu doses nke ọgwụ ka nwanyị dị ime No ọmụma dị. Ọzọkwa, e nweghị data na nwere mmetụta nke ọgwụ ọjọọ-antipsychotics na ụbụrụ nke nwa.

Ke ofụri ofụri, ahụ ike na-arụ ọrụ na-ahọrọ ghara iji "Sulpiride" maka ọgwụgwọ nke ime ndị inyom, ma e wezụga na mgbe ebe a mmetụta dị mma n'ihi na ndị inyom-enwe n'elu nwere ihe ize ndụ ka nke nwa ebu n'afọ. N'ọnọdụ dị otú ahụ, "Sulpiride" ntụziaka (reviews enyemaka n'ọrụ enen) aro ndinọ kasị ala-ekwe omume doses na ọ bụrụ na o kwere omume na-ebelata oge nke ọgwụgwọ.

Na mụrụ ụmụ na ụmụ nwaanyị na-ewere n'oge ime sulpiridsoderzhaschie ọgwụ mgbe ụfọdụ hụrụ eriri afọ mgbaàmà (bloating, na na. N.) Associated atropinopodobnye mmetụta nke neuroleptics. Mgbe ụfọdụ, i nwere ike ịnụ banyere extrapyramidal syndrome. N'oge ara welcome "sulpiride" contraindicated.

Mkpebi nke ọrịa "sulpiride"

Otutu nke ọrịa na ọgwụ ọjọọ, "Sulpiride" reviews doo a mma direction. Neuroleptic zuru ezu irè na ziri ezi na-kwuru, e ji mara. Ndị na-ewere "Sulpiride" ma ọ bụ ya analogues maka iche echiche mgbaàmà n'oge gastric ọnyá afọ ma ọ bụ duodenal ọnyá afọ, kọrọ a ọnụ ke siri nke abdominal mgbu na imeziwanye ihe na izugbe ọnọdụ.

Obere mpịakọta nke agwọ ọrịa (50 300 mg a ụbọchị) na-kenyere ka ọrịa na-anata na mkpesa nke Ugboro dizziness ịda dị iche iche ihe. Otutu n'ime ndị ọrịa bụ na afọ ojuju na-arụpụta nke ọgwụgwọ.

Large doses "sulpiride" (karịrị 600 mg kwa ụbọchị), na echiche nke ọgwụ na ahụ ike na-arụ ọrụ na-enye irè antipsychotic utịp ke ọrịa. Doses erughị 600 mg, na echiche nke ndị dọkịta na ndị ọrịa, na-ebu na-akpali akpali na antidepressant mmetụta.

E nwere otu ìgwè ndị ọrịa hapụrụ "sulpiride" na a na-ezighị ezi ụzọ. Otú ndị ịzụlite ọgbụgbọ, mkpali, giddiness. Na-adịghị mma mgbaàmà okụrede ke discontinuation nke "sulpiride".

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