Ahụ ike, Preparations
Omez - ntụziaka
Clinico-pharmacological Atiya ka nke bụ nke ọgwụ "Omez" - mgbochi ọnyá afọ mmadụ. A, na-emepụta na-emepụta a na-agwọ ya n'ụdị ike gelatin capsules uzo. On abụọ nke ntekwasa capsules e dere «OMEZ», na pụkwara enịm edenyere nke emeputa. The arọ nke otu Capsule bụ 20 milligrams. Capsules bụ ibe nke 10 mbak ọ bụla, na juru n'ọnụ ke katọn.
The n'ọrụ mgwa nke ọgwụ - omeprazole. N'okpuru a aha ya na-aha na nkwadebe njem. Ke adianade do, ụfọdụ na-emepụta na-emepụta ọgwụ bụ n'okpuru a aha. Adjuvants ekewet capsules bụ mannitol, lactose, ọcha talc, titanium dioxide, gelatin, sodium hydroxide, na sodium lauryl phosphate, sucrose.
The pharmacological edinam nke ọgwụ "Omez" ntụziaka ntuziaka na-akọwa na ndị na-esonụ ụzọ. Nke a antiulcer ọgwụ nwere ike inhibit ATP-ase na gastric mkpụrụ ndụ ma si otú na-arụ ọrụ na-egbochi ndị ikpeazụ nzọụkwụ nke usoro nke njikọ nke hydrochloric acid. N'ihi ya, e nwere a gụnyere ya ná ego nke kpaliri secretion. The isi iyi akpụ mkpali dịghị mkpa.
Mgbe e omeprazole amalite ngwa ngwa (ihe dị ka otu awa) na-eme ihe, na mmetụta ya nke ọma na-aga n'ihu ofụri usen.
Onye kasị ukwuu mmetụta nke ọgwụ ọjọọ, "Omez" ntụziaka na-ekpebi oge nke awa abụọ mgbe ingestion.
Ọ bụrụ na ọgwụ gosiri maka ọgwụgwọ nke ọnyá duodenum, na-arụsi ọrụ ike mgwa na-enye a Layer-3 intragastric onye Onyenwe anyị + nkeji iri na asa awa kasị dose of 20 mg. Iweghachi secretory ọrụ emee n'ime atọ ka ụbọchị ise.
The pharmacokinetic Njirimara nke ọgwụ "Omez" ntuziaka na-akọwa na ndị na-esonụ ụzọ. Absorption nke isi n'ọrụ mgwa omeprazole e ji ike na-pụtara ngwa ngwa etinye obi gị dum na eriri afọ tract. Mgbe ihe dị ka ọkara otu awa Cmax uru nke ọbara esịmde a kacha uru. Bioavailability "Omez" bụ banyere 30-40%.
Medicine "omeprazole" nwere a onwunwe na-emekọ ọma na plasma-edozi. nkịtị akara ruo 90%. N'ihi ya ọgwụ fọrọ nke nta kpamkpam metabolized na imeju mkpụrụ ndụ.
Oge nke ọgwụ bụ poluvyvoda oge n'etiti ọkara otu awa na mwepụ a rụrụ tumadi site na akụrụ ya. Ọ ga-iburu n'uche na na ikpe nke na-adịghị ala gbasara akụrụ odida ọnụego nke excretion nke ọgwụ mmiri na-ebelata hà na ọnụego nke ọnụ KK. The bioavailability nke ọgwụ dị elu na ndị agadi ndị ọrịa, na ọnụego nke excretion nke bekee n'okpuru. N'ihe banyere ọgwụ na ọrịa na hepatic ọdịda ọkara ndụ nke awa atọ na bioavailability bụ 100%.
Drug "Omez" ntụziaka ntuziaka tụrụ aro na-ewere na-mmiri mmiri, a Capsule kwesịrị iwere na a obere mmiri.
Ịnata ndidi dose na-ekenye a duodenal ọnyá afọ bụ 1 Capsule na 2-4 izu oge nke ochichi (n'ihi na-adịghị ala ala ọrịa ụdị). Na-eguzogide ọgwụ mgbe nwere ike ụba ruo 40 mg dose - 2 capsules a ụbọchị.
Maka ọgwụgwọ nke gastric ọnyá, nakwa dị ka erosive esophagitis ọnyá dose bụ 1-2 capsules kwa ụbọchị, na n'ikuku oge 4-8 izu. Duration nke eriri afọ ọnya na erosive na ọnyá agwa - 4-8 izu a kacha kwa ụbọchị dose nke 20 mg.
Bụrụ na nke ovadozu mgbaàmà ndị dị otú ahụ dị ka bịara ikiri ọhụụ, akọrọ ọnụ, ọgbụgbọ. Nnọọ adịkarịghị hụrụ arrhythmia, mgbagwoju anya na ụba agụụ.
Na ọgwụ ọgwụgwọ, "Omez" contraindications bụ: ọ gaghị ndinọ ka ụmụaka nakwa ndị inyom n'oge ime ma ọ bụ ara-udia a nwa. Tupu iji, nlezianya na-agụ ihe ndị mejupụtara nke ọgwụ na ewepu-ekwe omume nke mmetụta bụrụ na nke hypersensitivity ka ya mmiri.
Nkwadebe "Omez" ịchekwa na okpomọkụ agaghị elu karịa 25 Celsius C. Medicine dabara maka ojiji na nnabata na iwu nke nchekwa maka 3 afọ. The ọgwụ na-eresị naanị site ọgwụ.
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